Preparation and biological evaluation of indole, benzimidazole, and thienopyrrole piperazine carboxamides: potent human histamine h(4) antagonists.
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International Union of Basic and Clinical Pharmacology. XCVIII. Histamine ReceptorsNovel inhibitors of neurotropic alphavirus replication that improve host survival in a mouse model of acute viral encephalitis.Histamine H4 receptor antagonists as potent modulators of mammalian vestibular primary neuron excitability.The histamine H4 receptor in autoimmune disease.Molecular and biochemical pharmacology of the histamine H4 receptor.Histamine H4 receptor ligands and their potential therapeutic applications.Histamine H4 receptor ligands and their potential therapeutic applications: an update.Histamine H4 receptor ligands: future applications and state of art.Clinical Development of Histamine H4 Receptor Antagonists.Pharmacological Characterization of Human Histamine Receptors and Histamine Receptor Mutants in the Sf9 Cell Expression System.Effect of H4R antagonist N-(2-aminoethyl)-5-chloro-1H-indol-2-carboxamides and 5-chloro-2-(piperazin-1-ylmethyl)-1H-benzimidazole on histamine and 4-methylhistamine-induced mast cell response.Pharmacological characterization of the new histamine H4 receptor agonist VUF 8430.The histamine H4 receptor is functionally expressed on neurons in the mammalian CNSSynthetic FXR agonist GW4064 is a modulator of multiple G protein-coupled receptorsThe dual H3/4R antagonist thioperamide does not fully mimic the effects of the 'standard' H4R antagonist JNJ 7777120 in experimental murine asthma.N (α)-Methylated phenylhistamines exhibit affinity to the hH(4)R-a pharmacological and molecular modelling study.Pharmacological Characterization of 5-Substituted 1-[(2,3-dihydro-1-benzofuran-2-yl)methyl]piperazines: Novel Antagonists for the Histamine H3 and H4 Receptors with Anti-inflammatory Potential.1-[(2,3-Dihydro-1-benzofuran-2-yl) methyl]piperazines as novel anti-inflammatory compounds: Synthesis and evaluation on H3 R/H4 R.Biomass-Derived N-doped Carbon Materials with Silica-Supported Ultrasmall ZnO Nanoparticles: Robust Catalysts for the Green Synthesis of Benzimidazoles.10th anniversary Inflammation and Immune Diseases Drug Discovery and Development Summit. 20-21 March 2006, New Brunswick, USA.Role of the Histamine H4-Receptor in Bronchial Asthma.Molecular modeling and QSAR studies of a set of indole and benzimidazole derivatives as H₄ receptor antagonists.Mapping histamine H4receptor–ligand binding modes
P2860
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P2860
Preparation and biological evaluation of indole, benzimidazole, and thienopyrrole piperazine carboxamides: potent human histamine h(4) antagonists.
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2005 nî lūn-bûn
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2005年の論文
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2005年論文
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2005年論文
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2005年論文
@zh-hk
2005年論文
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2005年論文
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name
Preparation and biological eva ...... an histamine h(4) antagonists.
@en
type
label
Preparation and biological eva ...... an histamine h(4) antagonists.
@en
prefLabel
Preparation and biological eva ...... an histamine h(4) antagonists.
@en
P2093
P356
P1476
Preparation and biological eva ...... an histamine h(4) antagonists.
@en
P2093
Annette K Kwok
Barbara Pio
Chandra R Shah
Cheryl A Grice
Curt A Dvorak
James P Edwards
Jennifer D Venable
Jianmei Wei
Jill A Jablonowski
P304
P356
10.1021/JM0502081
P407
P577
2005-12-01T00:00:00Z