about
Design and pharmacological characterization of VUF14480, a covalent partial agonist that interacts with cysteine 98(3.36) of the human histamine H₄ receptor.The extracellular loop 2 (ECL2) of the human histamine H4 receptor substantially contributes to ligand binding and constitutive activity.The receptor concept in 3D: from hypothesis and metaphor to GPCR-ligand structures.Histamine H4 receptor ligands: future applications and state of art.Structure-based discovery and binding site analysis of histamine receptor ligands.Molecular Modelling Approaches for the Analysis of Histamine Receptors and Their Interaction with Ligands.Detailed analysis of biased histamine H₄ receptor signalling by JNJ 7777120 analogues.A structural chemogenomics analysis of aminergic GPCRs: lessons for histamine receptor ligand design.Structure-based virtual screening for fragment-like ligands of the G protein-coupled histamine H4 receptor
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Q34324177-A81C5E81-B550-48EF-82D1-C44953418B56Q35550563-4A1EB671-7746-4755-A613-DE145CF42B68Q38237899-1E2B79F1-22E5-422D-A23E-D52FE62033D2Q38250258-0CED2F56-3CD1-4E84-8F13-1A5D5AFABF49Q38972667-0698E12C-81DA-41BE-8FAD-BE8BD2E7D88AQ39007384-FEA5BF0B-4F16-4FD0-9E8F-BAB723AF6850Q39204577-0C0395CC-1900-4FAC-B2BA-99678168F969Q39411714-0261D0FE-E4F0-40EE-BEA6-506C23141018Q56991394-DE3817E4-13CD-4617-819A-31BE22E3FFE8
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description
im Januar 2013 veröffentlichter wissenschaftlicher Artikel
@de
wetenschappelijk artikel
@nl
наукова стаття, опублікована у 2013
@uk
name
Mapping histamine H4receptor–ligand binding modes
@en
Mapping histamine H4receptor–ligand binding modes
@nl
type
label
Mapping histamine H4receptor–ligand binding modes
@en
Mapping histamine H4receptor–ligand binding modes
@nl
prefLabel
Mapping histamine H4receptor–ligand binding modes
@en
Mapping histamine H4receptor–ligand binding modes
@nl
P2093
P2860
P50
P356
P1433
P1476
Mapping histamine H4receptor–ligand binding modes
@en
P2093
Eric E. J. Haaksma
Harald Engelhardt
Henry F. Vischer
Iwan J. P. de Esch
Sabine Schultes
P2860
P304
P356
10.1039/C2MD20212C
P577
2013-01-01T00:00:00Z