[Phe1psi(CH2-NH)Gly2]nociceptin-(1-13)-NH2 is an agonist of the nociceptin (ORL1) receptor.
about
Pharmacological profiles of a novel opioid receptor-like1 (ORL(1)) receptor antagonist, JTC-801Pharmacology of nociceptin and its receptor: a novel therapeutic targetComparison of the effects of [Phe1psi(CH2-NH)Gly2]nociceptin(1-13)NH2 in rat brain, rat vas deferens and CHO cells expressing recombinant human nociceptin receptorsCharacterization of opiates, neuroleptics, and synthetic analogs at ORL1 and opioid receptorsPharmacological properties of nociceptin/orphanin FQ-induced stimulation and inhibition of cyclic AMP formation in distinct layers of rat olfactory bulb[Phe1psi(CH2-NH)Gly2]nociceptin-(1 - 13)-NH2 activation of an inward rectifier as a partial agonist of ORL1 receptors in rat periaqueductal gray.Nociceptin, Phe(1)psi-nociceptin(1 - 13), nocistatin and prepronociceptin(154 - 181) effects on calcium channel currents and a potassium current in rat locus coeruleus in vitro.Activities of mixed NOP and mu-opioid receptor ligands.Central N/OFQ-NOP Receptor System in Pain Modulation.Pharmacological characterization of inhibitory effects of postsynaptic opioid and cannabinoid receptors on calcium currents in neonatal rat nucleus tractus solitariusNociceptin augments K(+) currents in hippocampal CA1 neurons by both ORL-1 and opiate receptor mechanisms.Characterization of the ORL(1) receptor on adrenergic nerves in the rat anococcygeus muscle.Characterization of [Nphe(1)]nociceptin(1-13)NH(2), a new selective nociceptin receptor antagonist.Nociceptin and the ORL-1 ligand [Phe1psi (CH2-NH)Gly2]nociceptin(1-13)NH2 exert anti-opioid effects in the Freund's adjuvant-induced arthritic rat model of chronic pain.Orphanin FQ/nociceptin and [Phe(1)Psi(CH(2)-NH)Gly(2)] nociceptin(1-13)-NH(2) stimulate gastric motor function in anaesthetized rats.Pre- and postsynaptic actions of opioid and orphan opioid agonists in the rat arcuate nucleus and ventromedial hypothalamus in vitro.
P2860
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P2860
[Phe1psi(CH2-NH)Gly2]nociceptin-(1-13)-NH2 is an agonist of the nociceptin (ORL1) receptor.
description
1998 nî lūn-bûn
@nan
1998年の論文
@ja
1998年論文
@yue
1998年論文
@zh-hant
1998年論文
@zh-hk
1998年論文
@zh-mo
1998年論文
@zh-tw
1998年论文
@wuu
1998年论文
@zh
1998年论文
@zh-cn
name
[Phe1psi(CH2-NH)Gly2]nocicepti ...... he nociceptin (ORL1) receptor.
@en
type
label
[Phe1psi(CH2-NH)Gly2]nocicepti ...... he nociceptin (ORL1) receptor.
@en
prefLabel
[Phe1psi(CH2-NH)Gly2]nocicepti ...... he nociceptin (ORL1) receptor.
@en
P2093
P1476
[Phe1psi(CH2-NH)Gly2]nocicepti ...... the nociceptin (ORL1) receptor
@en
P2093
J C Meunier
J L Butour
P356
10.1016/S0014-2999(98)00273-8
P407
P50
P577
1998-05-01T00:00:00Z