Synthesis and SAR of a novel metabotropic glutamate receptor 4 (mGlu4) antagonist: unexpected 'molecular switch' from a closely related mGlu4 positive allosteric modulator.
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Drugs for allosteric sites on receptors2013 Philip S. Portoghese Medicinal Chemistry Lectureship: drug discovery targeting allosteric sites.Development of allosteric modulators of GPCRs for treatment of CNS disordersRecent advances in the drug discovery of metabotropic glutamate receptor 4 (mGluR4) activators for the treatment of CNS and non-CNS disorders.Metabotropic glutamate receptor 4 (mGlu4)-positive allosteric modulators for the treatment of Parkinson's disease: historical perspective and review of the patent literature.Allosteric modulation of Class C GPCRs: a novel approach for the treatment of CNS disorders.Synthesis and SAR of substituted pyrazolo[1,5-a]quinazolines as dual mGlu(2)/mGlu(3) NAMs.
P2860
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P2860
Synthesis and SAR of a novel metabotropic glutamate receptor 4 (mGlu4) antagonist: unexpected 'molecular switch' from a closely related mGlu4 positive allosteric modulator.
description
2011 nî lūn-bûn
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2011年の論文
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2011年論文
@yue
2011年論文
@zh-hant
2011年論文
@zh-hk
2011年論文
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2011年論文
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2011年论文
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2011年论文
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2011年论文
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name
Synthesis and SAR of a novel m ...... positive allosteric modulator.
@en
Synthesis and SAR of a novel metabotropic glutamate receptor 4
@nl
type
label
Synthesis and SAR of a novel m ...... positive allosteric modulator.
@en
Synthesis and SAR of a novel metabotropic glutamate receptor 4
@nl
prefLabel
Synthesis and SAR of a novel m ...... positive allosteric modulator.
@en
Synthesis and SAR of a novel metabotropic glutamate receptor 4
@nl
P2093
P2860
P1476
Synthesis and SAR of a novel m ...... positive allosteric modulator.
@en
P2093
Corey R Hopkins
Dustin Haddenham
James M Salovich
Paige N Vinson
Rocio Zamorano
Thomas Utley
P2860
P304
P356
10.1016/J.BMCL.2011.09.131
P407
P577
2011-10-08T00:00:00Z