Dimers of class A G protein-coupled receptors function via agonist-mediated trans-activation of associated G proteins.
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Allostery at G protein-coupled receptor homo- and heteromers: uncharted pharmacological landscapesTrans-activation between 7TM domains: implication in heterodimeric GABAB receptor activationTASK Channels on Basal Forebrain Cholinergic Neurons Modulate Electrocortical Signatures of Arousal by HistamineTransmembrane domains of attraction on the TSH receptor.Requirements and ontology for a G protein-coupled receptor oligomerization knowledge base.The First Negative Allosteric Modulator for Dopamine D2 and D3 Receptors, SB269652 May Lead to a New Generation of Antipsychotic DrugsCell surface expression of alpha1D-adrenergic receptors is controlled by heterodimerization with alpha1B-adrenergic receptors.Monitoring the formation of dynamic G-protein-coupled receptor-protein complexes in living cells.The G protein-coupled receptor rhodopsin in the native membraneRhodopsin self-associates in asolectin liposomes.Allosteric signaling through an mGlu2 and 5-HT2A heteromeric receptor complex and its potential contribution to schizophreniaG protein-coupled receptor rhodopsin.Functional homomers and heteromers of dopamine D2L and D3 receptors co-exist at the cell surfaceRecent progress in alpha1-adrenergic receptor research.G Protein-coupled Receptor Biased Agonism.Heterodimerisation of G protein-coupled receptors: implications for drug design and ligand screening.Pathophysiology of GPCR Homo- and Heterodimerization: Special Emphasis on Somatostatin ReceptorsAllosteric communication between protomers of dopamine class A GPCR dimers modulates activation.Studies on the role of the receptor protein motifs possibly involved in electrostatic interactions on the dopamine D1 and D2 receptor oligomerization.CXCR2 chemokine receptor antagonism enhances DOP opioid receptor function via allosteric regulation of the CXCR2-DOP receptor heterodimer.Co-expression of mu and delta opioid receptors as receptor-G protein fusions enhances both mu and delta signalling via distinct mechanisms.Opsin oligomerization in a heterologous cell system.G protein activation by the leukotriene B4 receptor dimer. Evidence for an absence of trans-activation.Asymmetric conformational changes in a GPCR dimer controlled by G-proteins.Functional importance of a structurally distinct homodimeric complex of the family B G protein-coupled secretin receptor.Heterodimerization and surface localization of G protein coupled receptorsMepyramine, a histamine H1 receptor inverse agonist, binds preferentially to a G protein-coupled form of the receptor and sequesters G protein.Cooperative conformational changes in a G-protein-coupled receptor dimer, the leukotriene B(4) receptor BLT1.G-protein-coupled receptors: new approaches to maximise the impact of GPCRS in drug discovery.
P2860
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P2860
Dimers of class A G protein-coupled receptors function via agonist-mediated trans-activation of associated G proteins.
description
2003 nî lūn-bûn
@nan
2003年の論文
@ja
2003年学术文章
@wuu
2003年学术文章
@zh
2003年学术文章
@zh-cn
2003年学术文章
@zh-hans
2003年学术文章
@zh-my
2003年学术文章
@zh-sg
2003年學術文章
@yue
2003年學術文章
@zh-hant
name
Dimers of class A G protein-co ...... tion of associated G proteins.
@en
Dimers of class A G protein-co ...... tion of associated G proteins.
@nl
type
label
Dimers of class A G protein-co ...... tion of associated G proteins.
@en
Dimers of class A G protein-co ...... tion of associated G proteins.
@nl
prefLabel
Dimers of class A G protein-co ...... tion of associated G proteins.
@en
Dimers of class A G protein-co ...... tion of associated G proteins.
@nl
P2093
P2860
P356
P1476
Dimers of class A G protein-co ...... tion of associated G proteins.
@en
P2093
Graeme Milligan
John Pediani
Juan J Carrillo
P2860
P304
42578-42587
P356
10.1074/JBC.M306165200
P407
P577
2003-08-14T00:00:00Z