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Discovery and Optimization of a Selective Ligand for the Switch/Sucrose Nonfermenting-Related Bromodomains of Polybromo Protein-1 by the Use of Virtual Screening and Hydration AnalysisAn inhibitor-driven study for enhancing the selectivity of indirubin derivatives towards leishmanial Glycogen Synthase Kinase-3 over leishmanial cdc2-related protein kinase 3Identification of the substrate recognition and transport pathway in a eukaryotic member of the nucleobase-ascorbate transporter (NAT) familySoluble 3',6-substituted indirubins with enhanced selectivity toward glycogen synthase kinase -3 alter circadian period.Exploring and exploiting the systemic effects of deregulated replication licensing.Natural-Based Indirubins Display Potent Cytotoxicity toward Wild-Type and T315I-Resistant Leukemia Cell Lines.Synthesis, Docking Study and Kinase Inhibitory Activity of a Number of New Substituted Pyrazolo[3,4-c]pyridines.Roscovitine-derived, dual-specificity inhibitors of cyclin-dependent kinases and casein kinases 1.Novel Inverse Binding Mode of Indirubin Derivatives Yields Improved Selectivity for DYRK Kinases.Modeling, substrate docking, and mutational analysis identify residues essential for the function and specificity of a eukaryotic purine-cytosine NCS1 transporter.Structural basis for the synthesis of indirubins as potent and selective inhibitors of glycogen synthase kinase-3 and cyclin-dependent kinases.A substrate translocation trajectory in a cytoplasm-facing topological model of the monocarboxylate/H⁺ symporter Jen1p.Sesquiterpene lactones from Staehelina fruticosa.Combined Virtual and Experimental Screening for CK1 Inhibitors Identifies a Modulator of p53 and Reveals Important Aspects of in Silico Screening Performance.6-Br-5methylindirubin-3'oxime (5-Me-6-BIO) targeting the leishmanial glycogen synthase kinase-3 (GSK-3) short form affects cell-cycle progression and induces apoptosis-like death: exploitation of GSK-3 for treating leishmaniasis.NmeA, a novel efflux transporter specific for nucleobases and nucleosides, contributes to metal resistance in Aspergillus nidulans.Discovery of the glycogen phosphorylase-modulating activity of a resveratrol glucoside by using a virtual screening protocol optimized for solvation effects.Erratum to ‘Exploring and exploiting the systemic effects of deregulated replication licensing’ [Seminars in Cancer Biology 37–38C, (2016) 3–15]Novel indole–flutimide heterocycles with activity against influenza PA endonuclease and hepatitis C virusScreening of a composite library of clinically used drugs and well-characterized pharmacological compounds for cystathionine β-synthase inhibition identifies benserazide as a drug potentially suitable for repurposing for the experimental therapy ofDesign and synthesis of new C-nucleosides as potential adenosine deaminase inhibitorsSynthesis of 1,2-annulated adamantane heterocycles: structural determination studies of a bioactive cyclic sulfiteAn Integrated Computational Approach to the Phenomenon of Potent and Selective Inhibition of Aurora Kinases B and C by a Series of 7-Substituted IndirubinsTwo New Peltogynoids fromAcacia niloticaDelile with Kinase Inhibitory ActivityChemical Composition Of The Essential Oil OfCionura Erecta(Asclepiadaceae) Inforescences
P50
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P50
description
hulumtues
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հետազոտող
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Vassilios Myrianthopoulos
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Vassilios Myrianthopoulos
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Vassilios Myrianthopoulos
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Vassilios Myrianthopoulos
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Vassilios Myrianthopoulos
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Vassilios Myrianthopoulos
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Vassilios Myrianthopoulos
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Vassilios Myrianthopoulos
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Vassilios Myrianthopoulos
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Vassilios Myrianthopoulos
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prefLabel
Vassilios Myrianthopoulos
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Vassilios Myrianthopoulos
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Vassilios Myrianthopoulos
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Vassilios Myrianthopoulos
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Vassilios Myrianthopoulos
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P106
P1153
56162881700
P21
P31
P496
0000-0001-8359-9634