about
Structure-activity relationships of cyclic lactam analogues of alpha-melanocyte-stimulating hormone (alpha-MSH) targeting the human melanocortin-3 receptor60 YEARS OF POMC: Regulation of feeding and energy homeostasis by α-MSHNovel α-MSH analog causes weight loss in obese rats and minipigs and improves insulin sensitivitySolid-phase peptide head-to-side chain cyclodimerization: discovery of C(2)-symmetric cyclic lactam hybrid α-melanocyte-stimulating hormone (MSH)/agouti-signaling protein (ASIP) analogues with potent activities at the human melanocortin receptorsDevelopment of cyclic gamma-MSH analogues with selective hMC3R agonist and hMC3R/hMC5R antagonist activities.Melanocortin control of energy balance: evidence from rodent models.Effects of macrocycle size and rigidity on melanocortin receptor-1 and -5 selectivity in cyclic lactam alpha-melanocyte-stimulating hormone analogs.The melanocortin-4 receptor: physiology, pharmacology, and pathophysiology.Systematic Backbone Conformational Constraints on a Cyclic Melanotropin Ligand Leads to Highly Selective Ligands for Multiple Melanocortin Receptors.Substitution of arginine with proline and proline derivatives in melanocyte-stimulating hormones leads to selectivity for human melanocortin 4 receptor.Pro-Opiomelanocortin (POMC) Neurones, POMC-Derived Peptides, Melanocortin Receptors and Obesity: How Understanding of this System has Changed Over the Last Decade.Bench-top to clinical therapies: A review of melanocortin ligands from 1954 to 2016.Biological and conformational study of beta-substituted prolines in MT-II template: steric effects leading to human MC5 receptor selectivity.Orexigenic effect of the melanocortin MC4 receptor antagonist HS014 is inhibited only partially by neuropeptide Y Y1 receptor selective antagonists.Melanocortin receptors: new opportunities in drug discovery
P2860
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P2860
description
1986 nî lūn-bûn
@nan
1986年の論文
@ja
1986年学术文章
@wuu
1986年学术文章
@zh
1986年学术文章
@zh-cn
1986年学术文章
@zh-hans
1986年学术文章
@zh-my
1986年学术文章
@zh-sg
1986年學術文章
@yue
1986年學術文章
@zh-hant
name
Corticotropin inhibits food intake in rats.
@en
Corticotropin inhibits food intake in rats.
@nl
type
label
Corticotropin inhibits food intake in rats.
@en
Corticotropin inhibits food intake in rats.
@nl
prefLabel
Corticotropin inhibits food intake in rats.
@en
Corticotropin inhibits food intake in rats.
@nl
P1433
P1476
Corticotropin inhibits food intake in rats
@en
P2093
A Bertolini
R Poggioli
P304
P356
10.1016/0143-4179(86)90091-0
P577
1986-02-01T00:00:00Z