The suramin analogue NF279 is a novel and potent antagonist selective for the P2X(1) receptor.
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Molecular and functional properties of P2X receptors--recent progress and persisting challengesPhysiological role for P2X1 receptors in renal microvascular autoregulatory behaviorDesensitization masks nanomolar potency of ATP for the P2X1 receptorLack of contribution of P2X receptors to neurally mediated vasoconstriction in the rabbit kidney in vivo.Pharmacochemistry of the platelet purinergic receptors.P2X-selective purinergic antagonists are strong inhibitors of HIV-1 fusion during both cell-to-cell and cell-free infection.Vascular smooth muscle cells from small human omental arteries express P2X1 and P2X4 receptor subunits.Activation and regulation of purinergic P2X receptor channelsNeuropharmacology of purinergic receptors in human submucous plexus: Involvement of P2X₁, P2X₂, P2X₃ channels, P2Y and A₃ metabotropic receptors in neurotransmissionRenal autoregulation in P2X1 knockout mice.Medicinal chemistry of adenosine, P2Y and P2X receptors.Uridine adenosine tetraphosphate induces contraction and relaxation in rat aorta.Purinergic dysregulation in pulmonary hypertensionThe P2X1 ion channel in platelet function.Heteromeric assembly of P2X subunits.The P2X1 receptor and platelet function.Expression of P2 Purinergic Receptors in Mesenchymal Stem Cells and Their Roles in Extracellular Nucleotide Regulation of Cell Functions.Mammalian P2X7 receptor pharmacology: comparison of recombinant mouse, rat and human P2X7 receptors.Development of a comprehensive set of P2 receptor pharmacological research compoundsFunctional evidence that ATP or a related purine is an inhibitory NANC neurotransmitter in the mouse jejunum: study on the identity of P2X and P2Y purinoceptors involved.Exocytosis of ATP from astrocytes modulates phasic and tonic inhibition in the neocortex.Purinoreceptor-mediated current in myocytes from renal resistance arteries.Quantal release of ATP in mouse cortex.Interaction between cannabinoid CB1 receptors and endogenous ATP in the control of spontaneous mechanical activity in mouse ileum.Antagonism of P2X3-containing channels: commentary on Spelta et al.Calcium signaling pathways utilized by P2X receptors in freshly isolated preglomerular MVSMC.Ionotropic P2X purinoreceptors mediate synaptic transmission in rat pyramidal neurones of layer II/III of somato-sensory cortex.Effects of acute administration of and tachyphylaxis to alpha,beta-methylene ATP in the guinea-pig small intestine.Interaction of Purinergic P2X4 and P2X7 Receptor Subunits.Different mechanisms of hydroxyl radical production susceptible to purine P2 receptor antagonists between carbon monoxide poisoning and exogenous ATP in rat striatum.Involvement of P2X(7) purinergic receptor and MEK1/2 in interleukin-8 up-regulation by LL-37 in human gingival fibroblasts.
P2860
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P2860
The suramin analogue NF279 is a novel and potent antagonist selective for the P2X(1) receptor.
description
2000 nî lūn-bûn
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2000年の論文
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2000年学术文章
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2000年学术文章
@zh
2000年学术文章
@zh-cn
2000年学术文章
@zh-hans
2000年学术文章
@zh-my
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@zh-hant
name
The suramin analogue NF279 is a novel and potent antagonist selective for the P2X
@nl
The suramin analogue NF279 is ...... ctive for the P2X(1) receptor.
@en
type
label
The suramin analogue NF279 is a novel and potent antagonist selective for the P2X
@nl
The suramin analogue NF279 is ...... ctive for the P2X(1) receptor.
@en
prefLabel
The suramin analogue NF279 is a novel and potent antagonist selective for the P2X
@nl
The suramin analogue NF279 is ...... ctive for the P2X(1) receptor.
@en
P2093
P1433
P1476
The suramin analogue NF279 is ...... ctive for the P2X(1) receptor.
@en
P2093
P304
P356
10.1016/S0028-3908(00)00022-8
P577
2000-08-01T00:00:00Z