Biological profiles of highly potent novel endothelin antagonists selective for the ETA receptor.
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Characterization of endothelin receptors in the human umbilical artery and veinEndothelinEndothelin receptors and their antagonistsRole of endothelin in cardiovascular diseaseEndothelin@25 - new agonists, antagonists, inhibitors and emerging research frontiers: IUPHAR Review 12Pharmacology of a non-selective ETA and ETB receptor antagonist, TAK-044 and the inhibition of myocardial infarct size in rats[125I]-PD151242: a selective radioligand for human ETA receptorsAortic arch malformations and ventricular septal defect in mice deficient in endothelin-1Differential effects of endothelin on activation of renal mechanosensory nerves: stimulatory in high-sodium diet and inhibitory in low-sodium dietHuman big-endothelin-1 and endothelin-1 release prostacyclin via the activation of ET1 receptors in the rat perfused lungEvidence from receptor antagonists of an important role for ETB receptor-mediated vasoconstrictor effects of endothelin-1 in the rat kidney.Mediation via different receptors of the vasoconstrictor effects of endothelins and sarafotoxins in the systemic circulation and renal vasculature of the anaesthetized ratDiscrimination between ETA- and ETB-receptor-mediated effects of endothelin-1 and [Ala1,3,11,15]endothelin-1 by BQ-123 in the anaesthetized rat.Transcriptional down-regulation of the rabbit pulmonary artery endothelin B receptor during phenotypic modulationEndothelins and their inhibition in the human skin microcirculation: ET[1-31], a new vasoconstrictor peptide.Increased endothelin-1 production in fibroblasts derived from patients with systemic sclerosis.Stimuli of sensory-motor nerves terminate arterial contractile effects of endothelin-1 by CGRP and dissociation of ET-1/ET(A)-receptor complexesRole of mucosal blood flow: a conceptional review in gastric mucosal injury and protection.Endothelin-A receptor antagonism attenuates carcinoma-induced pain through opioids in mice.Activation of endothelin A receptors contributes to impaired responsiveness of renal mechanosensory nerves in congestive heart failureReversal of postischemic acute renal failure with a selective endothelinA receptor antagonist in the ratPhysiologic characterization of endothelin A and B receptor activity in the ovine fetal pulmonary circulationGene expression, localization, and characterization of endothelin A and B receptors in the human adrenal cortex.Modulation by endothelin-1 of spontaneous activity and membrane currents of atrioventricular node myocytes from the rabbit heart.Endothelin-1 and endothelin-3 regulate differently vasoconstrictor responses of smooth muscle of the porcine coronary artery.Endothelin ETA and ETB mRNA and receptors expressed by smooth muscle in the human vasculature: majority of the ETA sub-typeCharacterization of receptors mediating vascular responses to endothelin-1 in the conscious rat.Different endothelin receptors involved in endothelin-1- and sarafotoxin S6B-induced contractions of the human isolated coronary arteryBlock of endothelin-1-induced release of thromboxane A2 from the guinea pig lung and nitric oxide from the rabbit kidney by a selective ETB receptor antagonist, BQ-788Modulation of ET-1-induced contraction of human bronchi by airway epithelium-dependent nitric oxide release via ET(A) receptor activation.Endothelin-1-induced ET(A) receptor-mediated nociception, hyperalgesia and oedema in the mouse hind-paw: modulation by simultaneous ET(B) receptor activationEndotoxin causes up-regulation of endothelin receptors in cultured hepatic stellate cells via nitric oxide-dependent and -independent mechanisms.Pressor and pulmonary responses to ET-1(1-31) in guinea-pigs.Endothelin and endothelial dysfunction.Endothelin inhibits renin release from juxtaglomerular cells via endothelin receptors A and B via a transient receptor potential canonical-mediated pathway.Endothelin in the perinatal circulation.Biochemical and pharmacological profile of a potent and selective endothelin B-receptor antagonist, BQ-788.Endothelin-A-mediated vasoconstriction during exercise with advancing age.Enzymatic pathways involved in the generation of endothelin-1(1-31) from exogenous big endothelin-1 in the rabbit aorta.Endogenous endothelin maintains coronary artery tone by endothelin type A receptor stimulation in patients undergoing coronary arteriography.
P2860
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P2860
Biological profiles of highly potent novel endothelin antagonists selective for the ETA receptor.
description
1992 nî lūn-bûn
@nan
1992年の論文
@ja
1992年学术文章
@wuu
1992年学术文章
@zh-cn
1992年学术文章
@zh-hans
1992年学术文章
@zh-my
1992年学术文章
@zh-sg
1992年學術文章
@yue
1992年學術文章
@zh
1992年學術文章
@zh-hant
name
Biological profiles of highly ...... elective for the ETA receptor.
@en
Biological profiles of highly ...... elective for the ETA receptor.
@nl
type
label
Biological profiles of highly ...... elective for the ETA receptor.
@en
Biological profiles of highly ...... elective for the ETA receptor.
@nl
prefLabel
Biological profiles of highly ...... elective for the ETA receptor.
@en
Biological profiles of highly ...... elective for the ETA receptor.
@nl
P2093
P1433
P1476
Biological profiles of highly ...... elective for the ETA receptor.
@en
P2093
K Ishikawa
M Nishikibe
S Tsuchida
T Fukuroda
P304
P356
10.1016/0024-3205(92)90331-I
P407
P577
1992-01-01T00:00:00Z