about
Fragment-Based Discovery of 7-Azabenzimidazoles as Potent, Highly Selective, and Orally Active CDK4/6 InhibitorsFragment-Based Discovery of 6-Azaindazoles As Inhibitors of Bacterial DNA LigaseAllosteric inhibition of the neuropeptidase neurolysin.Efficient exploration of chemical space by fragment-based screening.Fragment-based approaches to the discovery of kinase inhibitors.Predicting "Hot" and "Warm" Spots for Fragment Binding.Fragment-Based Discovery of Potent and Selective DDR1/2 Inhibitors.Protein-ligand docking against non-native protein conformers.Discovery of novel inhibitors of Trypanosoma cruzi trans-sialidase from in silico screening.DNA gyrase (GyrB)/topoisomerase IV (ParE) inhibitors: synthesis and antibacterial activity.Fragment-to-Lead Medicinal Chemistry Publications in 2016.Docking performance of fragments and druglike compounds.Diverse, high-quality test set for the validation of protein-ligand docking performance.Fragment-to-Lead Medicinal Chemistry Publications in 2018Structure-Activity and Structure-Conformation Relationships of Aryl Propionic Acid Inhibitors of the Kelch-like ECH-Associated Protein 1/Nuclear Factor Erythroid 2-Related Factor 2 (KEAP1/NRF2) Protein-Protein InteractionFragment-to-Lead Medicinal Chemistry Publications in 2017
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P50
description
onderzoeker
@nl
researcher
@en
հետազոտող
@hy
name
Paul N. Mortenson
@ast
Paul N. Mortenson
@en
Paul N. Mortenson
@es
Paul N. Mortenson
@nl
Paul N. Mortenson
@sl
type
label
Paul N. Mortenson
@ast
Paul N. Mortenson
@en
Paul N. Mortenson
@es
Paul N. Mortenson
@nl
Paul N. Mortenson
@sl
prefLabel
Paul N. Mortenson
@ast
Paul N. Mortenson
@en
Paul N. Mortenson
@es
Paul N. Mortenson
@nl
Paul N. Mortenson
@sl
P106
P1153
6602760954
P21
P31
P496
0000-0002-3583-3163