Translocation of arrestin induced by human A(3) adenosine receptor ligands in an engineered cell line: comparison with G protein-dependent pathways
about
Seven transmembrane receptors as shapeshifting proteins: the impact of allosteric modulation and functional selectivity on new drug discovery.Probing biased/partial agonism at the G protein-coupled A(2B) adenosine receptor.Structure-based approaches to ligands for G-protein-coupled adenosine and P2Y receptors, from small molecules to nanoconjugates.Functionally biased modulation of A(3) adenosine receptor agonist efficacy and potency by imidazoquinolinamine allosteric enhancersAllosteric interactions across native adenosine-A3 receptor homodimers: quantification using single-cell ligand-binding kinetics.Pharmacological and therapeutic effects of A3 adenosine receptor agonistsFunctional selectivity of adenosine A1 receptor ligands?Therapeutic potential of β-arrestin- and G protein-biased agonists.Allosteric modulation and functional selectivity of G protein-coupled receptors.Structure-Activity Analysis of Biased Agonism at the Human Adenosine A3 Receptor.New paradigms in GPCR drug discovery.Novel 2- and 4-substituted 1H-imidazo[4,5-c]quinolin-4-amine derivatives as allosteric modulators of the A3 adenosine receptorFunctional selectivity of adenosine receptor ligandsProbing heterotrimeric G protein activation: applications to biased ligands.Effect of a toggle switch mutation in TM6 of the human adenosine A₃ receptor on Gi protein-dependent signalling and Gi-independent receptor internalization.Distinct Signaling Patterns of Allosteric Antagonism at the P2Y1 Receptor.
P2860
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P2860
Translocation of arrestin induced by human A(3) adenosine receptor ligands in an engineered cell line: comparison with G protein-dependent pathways
description
2008 nî lūn-bûn
@nan
2008 թուականի Ապրիլին հրատարակուած գիտական յօդուած
@hyw
2008 թվականի ապրիլին հրատարակված գիտական հոդված
@hy
2008年の論文
@ja
2008年論文
@yue
2008年論文
@zh-hant
2008年論文
@zh-hk
2008年論文
@zh-mo
2008年論文
@zh-tw
2008年论文
@wuu
name
Translocation of arrestin indu ...... h G protein-dependent pathways
@ast
Translocation of arrestin indu ...... h G protein-dependent pathways
@en
Translocation of arrestin indu ...... h G protein-dependent pathways
@nl
type
label
Translocation of arrestin indu ...... h G protein-dependent pathways
@ast
Translocation of arrestin indu ...... h G protein-dependent pathways
@en
Translocation of arrestin indu ...... h G protein-dependent pathways
@nl
prefLabel
Translocation of arrestin indu ...... h G protein-dependent pathways
@ast
Translocation of arrestin indu ...... h G protein-dependent pathways
@en
Translocation of arrestin indu ...... h G protein-dependent pathways
@nl
P2860
P1476
Translocation of arrestin indu ...... h G protein-dependent pathways
@en
P2860
P304
P356
10.1016/J.PHRS.2008.02.008
P407
P577
2008-03-08T00:00:00Z