An overview of the synthetic routes to the best selling drugs containing 6-membered heterocycles
about
Computational prediction and validation of an expert's evaluation of chemical probesVisible light mediated intermolecular [3 + 2] annulation of cyclopropylanilines with alkynes.Mild Pd-catalyzed aminocarbonylation of (hetero)aryl bromides with a palladacycle precatalystBenzo[b]quinolizinium Derivatives Have a Strong Antimalarial Activity and Inhibit Indoleamine Dioxygenase.Synthesis of High-Load, Hybrid Silica-Immobilized Heterocyclic Benzyl Phosphate (Si-OHBP) and Triazolyl Phosphate (Si-OHTP) Alkylating ReagentsChemoselective Palladium-Catalyzed Deprotonative Arylation/[1,2]-Wittig Rearrangement of Pyridylmethyl Ethers.Palladium-Catalyzed Benzylic C-H Arylation of Azaarylmethylamines.Palladium-Catalyzed Benzylic Arylation of Pyridylmethyl Silyl Ethers: One-Pot Synthesis of Aryl(pyridyl)methanols.A convenient route to symmetrically and unsymmetrically substituted 3,5-diaryl-2,4,6-trimethylpyridines via Suzuki-Miyaura cross-coupling reaction.Direct Assembly of Prenylated Heteroarenes through a Cascade Minisci Reaction/Dehydration Sequence.Transition metal-free one-pot synthesis of nitrogen-containing heterocycles.Design and synthesis of some new 2,3'-bipyridine-5-carbonitriles as potential anti-inflammatory/antimicrobial agents.Ionization of pyridine: Interplay of orbital relaxation and electron correlation.Modern advances in heterocyclic chemistry in drug discovery.NMR detection in biofluid extracts at sub-μM concentrations via para-H2 induced hyperpolarization.A Benzimidazole Proton Pump Inhibitor Increases Growth and Tolerance to Salt Stress in TomatoSyntheses of 3,4- and 1,4-dihydroquinazolines from 2-aminobenzylamine.Transetherification of 2,4-dimethoxynitrobenzene by aromatic nucleophilic substitution.Microwave-assisted cyclizations promoted by polyphosphoric acid esters: a general method for 1-aryl-2-iminoazacycloalkanes.Synthesis of Diverse (11)C-Labeled PET Radiotracers via Direct Incorporation of [(11)C]CO2.Ynamide carbopalladation: a flexible route to mono-, bi- and tricyclic azacycles.Synthetic versatility of 2-substituted-6-methyl 2,3-dihydropyridinones in the synthesis of polyfunctional piperidine-based compounds and related β amino acid derivatives.Synthesis of meta-Functionalized Pyridines by Selective Dehydrogenative Heterocondensation of β- and γ-Amino Alcohols.Rhodium-Catalyzed Asymmetric N-H Functionalization of Quinazolinones with Allenes and Allylic Carbonates: The First Enantioselective Formal Total Synthesis of (-)-Chaetominine.Inversion of cpADH5 Enantiopreference and Altered Chain Length Specificity for Methyl 3-Hydroxyalkanoates.Efficient Synthesis of 1,9-Substituted Benzo[h][1,6]naphthyridin-2(1H)-ones and Evaluation of their Plasmodium falciparum Gametocytocidal Activities.Rotational spectra of two six-membered heterocyclic N-methyl-piperidinol compounds: Conformations by OH rotation, N-methyl inversion, and ring puckering.Separation of structurally related primary aliphatic amines using hydrophilic interaction chromatography with fluorescence detection after postcolumn derivatization with o-phthaldialdehyde/mercaptoethanol.Trichloromethylthiolation of N-Heterocycles: Practical and Completely Regioselective.Mechanism and Scope of Base-Controlled Catalyst-Free N-Arylation of Amines with Unactivated Fluorobenzenes.An efficient and green reaction of isatins, 3-amino-1-phenyl-2-pyrazolin-5-one (3-amine-1H-pyrazole), and β-diketone in aqueous medium.Domino reaction of cyclic sulfamidate imines with Morita-Baylis-Hillman acetates promoted by DABCO: a metal-free approach to functionalized nicotinic acid derivatives.Carbodiimide insertion into sulfonimides: one-step route to azepine derivatives via a two-atom saccharin ring expansion.A Palladium(II)-Catalyzed C-H Activation Cascade Sequence for Polyheterocycle Formation.Enantioselective Aza Michael-Type Addition to Alkenyl Benzimidazoles Catalyzed by a Chiral Phosphoric Acid.Generic HPLC platform for automated enzyme reaction monitoring: Advancing the assay toolbox for transaminases and other PLP-dependent enzymes.Palladium-catalyzed carbonylative coupling of (2-azaaryl)methyl anion equivalents with (hetero)aryl bromides.A Convenient Late-Stage Fluorination of Pyridylic C-H Bonds with N-Fluorobenzenesulfonimide.In situ epoxide generation by dimethyldioxirane oxidation and the use of epichlorohydrin in the flow synthesis of a library of β-amino alcohols.Gold-catalyzed formal [4π + 2π]-cycloadditions of propiolate derivatives with unactivated nitriles.
P2860
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P2860
An overview of the synthetic routes to the best selling drugs containing 6-membered heterocycles
description
2013 nî lūn-bûn
@nan
2013 թուականի Հոկտեմբերին հրատարակուած գիտական յօդուած
@hyw
2013 թվականի հոտեմբերին հրատարակված գիտական հոդված
@hy
2013年の論文
@ja
2013年論文
@yue
2013年論文
@zh-hant
2013年論文
@zh-hk
2013年論文
@zh-mo
2013年論文
@zh-tw
2013年论文
@wuu
name
An overview of the synthetic r ...... aining 6-membered heterocycles
@ast
An overview of the synthetic r ...... aining 6-membered heterocycles
@en
An overview of the synthetic r ...... aining 6-membered heterocycles
@nl
type
label
An overview of the synthetic r ...... aining 6-membered heterocycles
@ast
An overview of the synthetic r ...... aining 6-membered heterocycles
@en
An overview of the synthetic r ...... aining 6-membered heterocycles
@nl
prefLabel
An overview of the synthetic r ...... aining 6-membered heterocycles
@ast
An overview of the synthetic r ...... aining 6-membered heterocycles
@en
An overview of the synthetic r ...... aining 6-membered heterocycles
@nl
P2860
P356
P1476
An overview of the synthetic r ...... aining 6-membered heterocycles
@en
P2860
P304
P356
10.3762/BJOC.9.265
P407
P577
2013-10-30T00:00:00Z