Application of palladium-mediated (18)F-fluorination to PET radiotracer development: overcoming hurdles to translation. - Test2 - elhamkhani - TriplyDB

Application of palladium-mediated (18)F-fluorination to PET radiotracer development: overcoming hurdles to translation.

Application of palladium-mediated (18)F-fluorination to PET radiotracer development: overcoming hurdles to translation.

http://www.wikidata.org/entity/Q31114482

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A philosophy for CNS radiotracer design Late-Stage Fluorination: From Fundamentals to Application Synthesis and evaluation of 4-[18F]fluoropropoxy-3-iodobenzylguanidine ([18F]FPOIBG): A novel 18F-labeled analogue of MIBG.Titania-catalyzed radiofluorination of tosylated precursors in highly aqueous medium.18F-Fluoroform: a 18F-trifluoromethylating agent for the synthesis of SCF218F-aromatic derivatives.A Transmetalation Reaction Enables the Synthesis of [18F]5-Fluorouracil from [18F]Fluoride for Human PET Imaging Late-stage formation of carbon-fluorine bonds.Current radiosynthesis strategies for 5-HT2A receptor PET tracers.Fluorination methods for drug discovery and development.Fluorine-18 patents (2009-2015). Part 2: new radiochemistry.Fluorine-18 labelled building blocks for PET tracer synthesis.Sulfonium salts as leaving groups for aromatic labelling of drug-like small molecules with fluorine-18.Copper-catalyzed [18F]fluorination of (mesityl)(aryl)iodonium salts.18F-Deoxyfluorination of Phenols via Ru π-Complexes Late-stage [(18)F]Fluorination: New Solutions to Old Problems Mechanism of Electrophilic Fluorination with Pd(IV): Fluoride Capture and Subsequent Oxidative Fluoride Transfer(.)Anion-Dependent Switch in C-X Reductive Elimination Diastereoselectivity.Moving Metal-Mediated (18)F-Fluorination from Concept to Clinic.Synthesis of [18F]Arenes via the Copper-Mediated [18F]Fluorination of Boronic Acids.Synthesis of [18 F]Fluoroarenes by Nucleophilic Radiofluorination of N-Arylsydnones.Alcohol-Enhanced Cu-Mediated Radiofluorination.Copper-mediated aromatic radiofluorination revisited: efficient production of PET tracers on a preparative scale.Enhanced copper-mediated (18)F-fluorination of aryl boronic esters provides eight radiotracers for PET applications.[(18) F]CuCF3 : a [(18) F]trifluoromethylating agent for arylboronic acids and aryl iodides.

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P2860

Application of palladium-mediated (18)F-fluorination to PET radiotracer development: overcoming hurdles to translation.

http://www.wikidata.org/entity/Q31114482

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2013 nî lūn-bûn

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2013 թվականի մարտին հրատարակված գիտական հոդված

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2013年の論文

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2013年論文

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2013年論文

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2013年論文

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2013年論文

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2013年论文

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Application of palladium-media ...... coming hurdles to translation.

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Application of palladium-media ...... coming hurdles to translation.

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Adam S Kamlet

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Christian K Moseley

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Eunsung Lee

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Nickeisha Stephenson

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Stephen M Carlin

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Tobias Ritter

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Jacob M. Hooker

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