Biological and conformational evaluation of bifunctional compounds for opioid receptor agonists and neurokinin 1 receptor antagonists possessing two penicillamines
about
Synthesis and biological evaluation of compact, conformationally constrained bifunctional opioid agonist - neurokinin-1 antagonist peptidomimetics.Discovery of tripeptide-derived multifunctional ligands possessing delta/mu opioid receptor agonist and neurokinin 1 receptor antagonist activities.Truncation of the peptide sequence in bifunctional ligands with mu and delta opioid receptor agonist and neurokinin 1 receptor antagonist activitiesNeurokinin 1 and opioid receptors: relationships and interactions in nervous system.In vivo antinociception of potent mu opioid agonist tetrapeptide analogues and comparison with a compact opioid agonist-neurokinin 1 receptor antagonist chimeraDual Alleviation of Acute and Neuropathic Pain by Fused Opioid Agonist-Neurokinin 1 Antagonist Peptidomimetics.Design of novel neurokinin 1 receptor antagonists based on conformationally constrained aromatic amino acids and discovery of a potent chimeric opioid agonist-neurokinin 1 receptor antagonist.
P2860
Q35107996-BC11DD8A-24C2-4647-9D52-6CD55726D0B7Q36274639-02722340-13C6-494E-BCB1-B59B884EBBA7Q37261127-3E952936-7F35-4FA6-9067-545387FB9B16Q38926264-832FE558-E99C-4B5E-9DEF-7FFF11A3A7FAQ41440337-E8690DA4-24C4-4A0F-81B5-35F710D65032Q42053439-ADFB9301-3537-424A-BF3F-D19B87AB87E1Q42735567-6632EDF5-636A-4023-9FBA-A2FD17919734
P2860
Biological and conformational evaluation of bifunctional compounds for opioid receptor agonists and neurokinin 1 receptor antagonists possessing two penicillamines
description
2010 nî lūn-bûn
@nan
2010 թուականի Օգոստոսին հրատարակուած գիտական յօդուած
@hyw
2010 թվականի օգոստոսին հրատարակված գիտական հոդված
@hy
2010年の論文
@ja
2010年論文
@yue
2010年論文
@zh-hant
2010年論文
@zh-hk
2010年論文
@zh-mo
2010年論文
@zh-tw
2010年论文
@wuu
name
Biological and conformational ...... possessing two penicillamines
@ast
Biological and conformational ...... possessing two penicillamines
@en
Biological and conformational ...... possessing two penicillamines
@nl
type
label
Biological and conformational ...... possessing two penicillamines
@ast
Biological and conformational ...... possessing two penicillamines
@en
Biological and conformational ...... possessing two penicillamines
@nl
prefLabel
Biological and conformational ...... possessing two penicillamines
@ast
Biological and conformational ...... possessing two penicillamines
@en
Biological and conformational ...... possessing two penicillamines
@nl
P2093
P2860
P356
P1476
Biological and conformational ...... possessing two penicillamines
@en
P2093
Edita Navratilova
Frank Porreca
Henry I Yamamura
Josephine Lai
Neil E Jacobsen
Padma Nair
Shou-Wu Ma
Takashi Yamamoto
Todd W Vanderah
P2860
P304
P356
10.1021/JM100157M
P407
P577
2010-08-01T00:00:00Z