Investigation of the binding and functional properties of extended length D3 dopamine receptor-selective antagonists
about
The First Negative Allosteric Modulator for Dopamine D2 and D3 Receptors, SB269652 May Lead to a New Generation of Antipsychotic DrugsTargeting the dopamine D3 receptor: an overview of drug design strategies.Norbenzomorphan Framework as a Novel Scaffold for Generating Sigma 2 Receptor/PGRMC1 Subtype-Selective LigandsNovel Analogues of (R)-5-(Methylamino)-5,6-dihydro-4H-imidazo[4,5,1-ij]quinolin-2(1H)-one (Sumanirole) Provide Clues to Dopamine D2/D3 Receptor Agonist Selectivity.Advances and challenges in the search for D2 and D3 dopamine receptor-selective compounds.Highly Selective Dopamine D3 Receptor (D3R) Antagonists and Partial Agonists Based on Eticlopride and the D3R Crystal Structure: New Leads for Opioid Dependence Treatment.The action of a negative allosteric modulator at the dopamine D2 receptor is dependent upon sodium ions.The E2.65A mutation disrupts dynamic binding poses of SB269652 at the dopamine D2 and D3 receptors.Synthesis and Pharmacological Characterization of Novel trans-Cyclopropylmethyl-Linked Bivalent Ligands That Exhibit Selectivity and Allosteric Pharmacology at the Dopamine D3 Receptor (D3R).
P2860
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P2860
Investigation of the binding and functional properties of extended length D3 dopamine receptor-selective antagonists
description
2014 nî lūn-bûn
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2014年の論文
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2014年論文
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2014年論文
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2014年論文
@zh-hk
2014年論文
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2014年論文
@zh-tw
2014年论文
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2014年论文
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name
Investigation of the binding a ...... receptor-selective antagonists
@ast
Investigation of the binding a ...... receptor-selective antagonists
@en
type
label
Investigation of the binding a ...... receptor-selective antagonists
@ast
Investigation of the binding a ...... receptor-selective antagonists
@en
prefLabel
Investigation of the binding a ...... receptor-selective antagonists
@ast
Investigation of the binding a ...... receptor-selective antagonists
@en
P2093
P2860
P1476
Investigation of the binding a ...... receptor-selective antagonists
@en
P2093
Amy E Moritz
Ashwini K Banala
Brittney N Miller
Cheryse A Furman
Christopher D Sibley
David R Sibley
Noel M Paul
R Benjamin Free
Rebecca A Roof
Trevor B Doyle
P2860
P304
P356
10.1016/J.EURONEURO.2014.11.013
P407
P577
2014-11-29T00:00:00Z