Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction
about
Polyacetylenes from Notopterygium incisum--new selective partial agonists of peroxisome proliferator-activated receptor-gammaSlow receptor dissociation kinetics differentiate macitentan from other endothelin receptor antagonists in pulmonary arterial smooth muscle cellsPhase I hydroxylated metabolites of the K2 synthetic cannabinoid JWH-018 retain in vitro and in vivo cannabinoid 1 receptor affinity and activityPrKX is a novel catalytic subunit of the cAMP-dependent protein kinase regulated by the regulatory subunit type IChloroform extract of hog barn dust modulates skeletal muscle ryanodine receptor calcium-release channel (RyR1)Peroxidase activity and structural transitions of cytochrome c bound to cardiolipin-containing membranesIdentification and characterization of two G protein-coupled receptors for neuropeptide FFToward selective drug development for the human 5-hydroxytryptamine 1E receptor: a comparison of 5-hydroxytryptamine 1E and 1F receptor structure-affinity relationshipsThe Kell protein of the common K2 phenotype is a catalytically active metalloprotease, whereas the rare Kell K1 antigen is inactive. Identification of novel substrates for the Kell proteinPro-urokinase-type plasminogen activator is a substrate for hepsinSelective and ATP-dependent translocation of peptides by the homodimeric ATP binding cassette transporter TAP-like (ABCB9)Solution structure and mutational analysis of pituitary adenylate cyclase-activating polypeptide binding to the extracellular domain of PAC1-RSAntidepressant- and cocaine-sensitive human serotonin transporter: molecular cloning, expression, and chromosomal localizationIdentification of a novel hypothalamic neuropeptide Y receptor associated with feeding behaviorAtypical responsiveness of the orphan receptor GPR55 to cannabinoid ligandsCloning of another human serotonin receptor (5-HT1F): a fifth 5-HT1 receptor subtype coupled to the inhibition of adenylate cyclaseThe human proton-coupled folate transporter (hPCFT): modulation of intestinal expression and function by drugsGalanin pathogenic mutations in temporal lobe epilepsyDeveloping dual and specific inhibitors of dimethylarginine dimethylaminohydrolase-1 and nitric oxide synthase: toward a targeted polypharmacology to control nitric oxideStable expression of human H1-histamine-receptor cDNA in Chinese hamster ovary cells. Pharmacological characterisation of the protein, tissue distribution of messenger RNA and chromosomal localisation of the geneActivation of 5-HT1A receptors expressed in NIH-3T3 cells induces focus formation and potentiates EGF effect on DNA synthesisMolecular characterization of the mouse beta 3-adrenergic receptor: relationship with the atypical receptor of adipocytesHuman serotonin 1D receptor is encoded by a subfamily of two distinct genes: 5-HT1D alpha and 5-HT1D betaThe enzyme-activated irreversible inhibition of type-B monoamine oxidase by 3-(4-[(3-chlorophenyl)methoxy]phenyl)-5-[(methylamino) methyl]-2-oxazolidinone methanesulphonate (compound MD 780236) and the enzyme-catalysed oxidation of this compound asDiscovery and characterization of vicriviroc (SCH 417690), a CCR5 antagonist with potent activity against human immunodeficiency virus type 1Heterozygous alpha 2A-adrenergic receptor mice unveil unique therapeutic benefits of partial agonists.Ethanol potently and competitively inhibits binding of the alcohol antagonist Ro15-4513 to alpha4/6beta3delta GABAA receptorsStructural requirements of ligands for the oxysterol liver X receptors LXRalpha and LXRbetaMolecular cloning, characterization, and localization of a high-affinity serotonin receptor (5-HT7) activating cAMP formationSoluble type II interleukin 1 (IL-1) receptor binds and blocks processing of IL-1 beta precursor and loses affinity for IL-1 receptor antagonistIsolation of cDNAs for two distinct human Fc receptors by ligand affinity cloningMolecular cloning and characterization of the human A3 adenosine receptor.Blockage of 5HT2C serotonin receptors by fluoxetine (Prozac)Jasmonate perception by inositol-phosphate-potentiated COI1-JAZ co-receptorMicrobial ureases: significance, regulation, and molecular characterizationTargeted mutations of Bacillus anthracis dihydrofolate reductase condense complex structure−activity relationshipsThe structural basis for agonist and partial agonist action on a β(1)-adrenergic receptorSUMO protease SENP1 induces isomerization of the scissile peptide bondCharacterization and distribution of alpha 2-adrenergic receptors in the human intestinal mucosaMarine algal toxin azaspiracid is an open-state blocker of hERG potassium channels
P2860
Q21090765-1E3B1AE3-92ED-4E16-8B02-EC579869E927Q21133932-E7CFCA71-EF28-41D3-9CC2-AAEFE3179FE5Q21135310-99ED3F21-869D-4A23-9E55-643E686A8AE5Q22008785-8D82D30E-A9EF-431E-B016-9F39B9A4A8EDQ23911039-8C3A09D4-44FF-4BD2-9CE5-48D5CE71B08AQ23918788-873CC889-0B46-477C-A34C-08144B5BC636Q24290374-51199CA9-AF7D-4401-97EF-4DD4EE838FFAQ24297642-698CE188-F23D-49B8-B9C9-2505344E8F36Q24298076-E338C38F-1FAC-4812-B324-7EBF2DE301B8Q24299743-045E96B8-1830-40C5-8F12-564AC45F4DE6Q24301098-72306164-11C1-4F2C-9205-FEA8E647C971Q24304303-DC023598-ECC9-4514-8057-E0C607EFF852Q24308751-CF5B1FF9-F23F-4FE5-9CEA-E65D86F590D3Q24309148-C8082824-9581-4EEA-A8C9-B8B9F65D1815Q24311776-32A90749-68AF-46B4-AF8D-397134CD7F56Q24313646-F68282B3-ACA4-4B74-AEB3-82C0FF2F1872Q24317138-7B987B80-2BD0-4EAF-8554-18B1D26C6355Q24319705-7F6A2329-1C01-44D7-B64E-8AFBB912F74DQ24321779-5CF7C064-6A1D-40D4-B12F-143A1D88FA37Q24322039-4C4F94EF-B498-45A2-B9CA-5CBAA2471173Q24337397-DD9E7DB4-0C37-4B81-B027-9F1227CBD534Q24338133-12E57BF6-B504-43E5-9AE0-66BA4BD781D9Q24338360-47B32530-BE6C-46F6-95C2-82F99E7EF40CQ24530005-A16DF2B4-82E6-4F5D-952A-09531F6A75FFQ24534620-56E935A9-12BB-4C35-8A6D-DCF6D7EC9422Q24535863-476EBA7B-7027-40B9-A7FD-362D9E8DE4E5Q24548490-E9B38977-4E1E-4F81-B19C-FA8E1985E4A8Q24553340-01FF9255-8E7D-497B-B19E-9AA0C17B6CF7Q24561553-0169BB7A-F7BF-4C2F-90E6-B34DD9D3AE74Q24563274-8B29ECAE-F4FC-44EF-9801-5511FF113FE3Q24564255-E67FF2FC-1B45-4301-85BF-92F97756C747Q24564442-737EB6E3-6E0A-40E1-9901-8406333D7CDFQ24564795-6822CF1C-3969-4B30-8563-66F2FAEBDB80Q24569663-FF0B1D57-AFC3-4ACA-B22B-8DDBFA156EE7Q24594053-56DC7829-DB4B-4527-8002-20987EC4FE4EQ24594645-29B68B51-82E4-4D6D-9E24-2CAD49D20D5AQ24594844-42B35C95-3926-44EE-8258-6F659322C577Q24596746-6775603A-5DDE-4E4E-9788-58C04F3FED4BQ24598150-1F723A06-24D1-4F1A-A987-32E0B5D3D5F3Q24599453-0E0AD868-C824-438B-B9F1-EF4E1D0E8F59
P2860
Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction
description
1973 nî lūn-bûn
@nan
1973 թուականի Դեկտեմբերին հրատարակուած գիտական յօդուած
@hyw
1973 թվականի դեկտեմբերին հրատարակված գիտական հոդված
@hy
1973年の論文
@ja
1973年論文
@yue
1973年論文
@zh-hant
1973年論文
@zh-hk
1973年論文
@zh-mo
1973年論文
@zh-tw
1973年论文
@wuu
name
Relationship between the inhib ...... (I50) of an enzymatic reaction
@ast
Relationship between the inhib ...... (I50) of an enzymatic reaction
@en
Relationship between the inhib ...... (I50) of an enzymatic reaction
@nl
type
label
Relationship between the inhib ...... (I50) of an enzymatic reaction
@ast
Relationship between the inhib ...... (I50) of an enzymatic reaction
@en
Relationship between the inhib ...... (I50) of an enzymatic reaction
@nl
prefLabel
Relationship between the inhib ...... (I50) of an enzymatic reaction
@ast
Relationship between the inhib ...... (I50) of an enzymatic reaction
@en
Relationship between the inhib ...... (I50) of an enzymatic reaction
@nl
P3181
P1476
Relationship between the inhib ...... (I50) of an enzymatic reaction
@en
P2093
P304
P3181
P356
10.1016/0006-2952(73)90196-2
P407
P577
1973-12-01T00:00:00Z