about
Sub-picomolar relaxin signalling by a pre-assembled RXFP1, AKAP79, AC2, beta-arrestin 2, PDE4D3 complexAntagonists show GTP-sensitive high-affinity binding to the sigma-1 receptorRole of receptors in Bacillus thuringiensis crystal toxin activityCardiac cAMP: production, hydrolysis, modulation and detectionSuramin inhibits initiation of defense signaling by systemin, chitosan, and a beta-glucan elicitor in suspension-cultured Lycopersicon peruvianum cellsPhospholipid synthesis in yeast: regulation by phosphorylationCubozoan genome illuminates functional diversification of opsins and photoreceptor evolutionSuramin and the suramin analogue NF307 discriminate among calmodulin-binding sitesRegulation of amyloid precursor protein processing by serotonin signalingThe Suramin Derivative NF449 Interacts with the 5-fold Vertex of the Enterovirus A71 Capsid to Prevent Virus Attachment to PSGL-1 and Heparan SulfateA mechanism of cell death involving an adenylyl cyclase/PKA signaling pathway is induced by the Cry1Ab toxin of Bacillus thuringiensis.NF449 is a novel inhibitor of fibroblast growth factor receptor 3 (FGFR3) signaling active in chondrocytes and multiple myeloma cellsAntagonists of the receptor-G protein interface block Gi-coupled signal transduction.Identification of phosphotyrosine mimetic inhibitors of human tyrosyl-DNA phosphodiesterase I by a novel AlphaScreen high-throughput assayInduction of Galphas contributes to the paradoxical stimulation of cytosolic phospholipase A2alpha expression by cortisol in human amnion fibroblasts.ML290 is a biased allosteric agonist at the relaxin receptor RXFP1.Lipid metabolism and vesicle trafficking: more than just greasing the transport machinery.Resistance of macrophages to Mycobacterium avium is induced by alpha2-adrenergic stimulation.Chronic loss of noradrenergic tone produces β-arrestin2-mediated cocaine hypersensitivity and alters cellular D2 responses in the nucleus accumbensThe G protein α subunit Gαs is a tumor suppressor in Sonic hedgehog-driven medulloblastomaTime-Resolved Fluorescence Resonance Energy Transfer Assay for Discovery of Small-Molecule Inhibitors of Methyl-CpG Binding Domain Protein 2.Development of high throughput screening assays and pilot screen for inhibitors of metalloproteases meprin α and β.Activation and regulation of purinergic P2X receptor channelsAldosterone stimulates vacuolar H(+)-ATPase activity in renal acid-secretory intercalated cells mainly via a protein kinase C-dependent pathway.Tricyclic Antidepressant Amitriptyline-induced Glial Cell Line-derived Neurotrophic Factor Production Involves Pertussis Toxin-sensitive Gαi/o Activation in Astroglial Cells.Cardiac Effects of Attenuating Gsα - Dependent SignalingThe β2-adrenoceptor activates a positive cAMP-calcium feedforward loop to drive breast cancer cell invasion.Acylated and unacylated ghrelin impair skeletal muscle atrophy in mice.Signaling mechanism of HIV-1 gp120 and virion-induced IL-1beta release in primary human macrophages.GLP-2 Attenuates LPS-Induced Inflammation in BV-2 Cells by Inhibiting ERK1/2, JNK1/2 and NF-κB Signaling Pathways.An arrestin-dependent multi-kinase signaling complex mediates MIP-1beta/CCL4 signaling and chemotaxis of primary human macrophages.Inhibition of heterotrimeric G protein signaling by a small molecule acting on Galpha subunit.Molecular signaling underlying bulleyaconitine A (BAA)-induced microglial expression of prodynorphin.Probing heterotrimeric G protein activation: applications to biased ligands.Molecular targeting of Gα and Gβγ subunits: a potential approach for cancer therapeutics.Selectivity of pharmacological tools: implications for use in cell physiology. A review in the theme: Cell signaling: proteins, pathways and mechanisms.Wnt-5a/Frizzled9 Receptor Signaling through the Gαo-Gβγ Complex Regulates Dendritic Spine FormationA cell-permeable inhibitor to trap Gαq proteins in the empty pocket conformation.Suramin affects coupling of rhodopsin to transducin.Antagonism of endogenous putative P2Y receptors reduces the growth of MDCK-derived cysts cultured in vitro.
P2860
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P2860
description
1998 nî lūn-bûn
@nan
1998年の論文
@ja
1998年論文
@yue
1998年論文
@zh-hant
1998年論文
@zh-hk
1998年論文
@zh-mo
1998年論文
@zh-tw
1998年论文
@wuu
1998年论文
@zh
1998年论文
@zh-cn
name
Gsalpha-selective G protein antagonists.
@ast
Gsalpha-selective G protein antagonists.
@en
type
label
Gsalpha-selective G protein antagonists.
@ast
Gsalpha-selective G protein antagonists.
@en
prefLabel
Gsalpha-selective G protein antagonists.
@ast
Gsalpha-selective G protein antagonists.
@en
P2093
P2860
P356
P1476
Gsalpha-selective G protein antagonists.
@en
P2093
A Kreimeyer
M Freissmuth
M Waldhoer
P2860
P304
P356
10.1073/PNAS.95.1.346
P407
P577
1998-01-01T00:00:00Z