Steroidal scaffolds as FXR and GPBAR1 ligands: from chemistry to therapeutical application.
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Navigation in bile acid chemical space: discovery of novel FXR and GPBAR1 ligandsLigand binding to telomeric G-quadruplex DNA investigated by funnel-metadynamics simulations.Targeting Bile Acid Receptors: Discovery of a Potent and Selective Farnesoid X Receptor Agonist as a New Lead in the Pharmacological Approach to Liver Diseases.Blinded evaluation of farnesoid X receptor (FXR) ligands binding using molecular docking and free energy calculations.The crosstalk between gut microbiota and obesity and related metabolic disorders.Role of farnesoid X receptor in cholestasis.Insights on FXR selective modulation. Speculation on bile acid chemical space in the discovery of potent and selective agonists.Epoxide functionalization on cholane side chains in the identification of G-protein coupled bile acid receptor (GPBAR1) selective agonists
P2860
Q28831219-60DC5049-CE61-4E74-B6A5-2CDF0E5AE0EBQ37711622-B9D2D613-8B78-4DFF-BF72-83E26BFACBD7Q37727582-41F0E0CC-86CE-431E-9899-AC34B21CBEEAQ38597033-A2758C06-59BF-43F7-9B3C-5E4F02EF887BQ38837418-4C2A01DE-2A2D-40DF-9E68-6030221AB8EAQ38887864-DA265332-1D1A-4AC5-B4E8-824D7748C879Q43102009-32E47FB2-CD17-4758-88F5-82F5E003DDB6Q58861672-44C3B85A-8C0F-4725-B776-5B8FF7B63464
P2860
Steroidal scaffolds as FXR and GPBAR1 ligands: from chemistry to therapeutical application.
description
2015 nî lūn-bûn
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2015年の論文
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2015年論文
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2015年論文
@zh-hant
2015年論文
@zh-hk
2015年論文
@zh-mo
2015年論文
@zh-tw
2015年论文
@wuu
2015年论文
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2015年论文
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name
Steroidal scaffolds as FXR and ...... to therapeutical application.
@en
type
label
Steroidal scaffolds as FXR and ...... to therapeutical application.
@en
prefLabel
Steroidal scaffolds as FXR and ...... to therapeutical application.
@en
P2093
P2860
P356
P1476
Steroidal scaffolds as FXR and ...... to therapeutical application.
@en
P2093
Eleonora Distrutti
Stefano Fiorucci
Valentina Sepe
P2860
P304
P356
10.4155/FMC.15.54
P577
2015-07-01T00:00:00Z