Design, synthesis and biological evaluation of novel quinazoline derivatives as potential antitumor agents: molecular docking study.
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Identification of potent EGFR inhibitors from TCM Database@TaiwanModification, biological evaluation and 3D QSAR studies of novel 2-(1,3-diaryl- 4,5-dihydro-1H-pyrazol-5-yl)phenol derivatives as inhibitors of B-Raf kinaseAn Investigation of Molecular Docking and Molecular Dynamic Simulation on Imidazopyridines as B-Raf Kinase InhibitorsA Combined Pharmacophore Modeling, 3D QSAR and Virtual Screening Studies on Imidazopyridines as B-Raf InhibitorsVirtual screening of natural compounds as inhibitors of EGFR 696-1022 T790M associated with non-small cell lung cancerAdvances in the design and synthesis of prazosin derivatives over the last ten years.Synthesis and biological evaluation of benzimidazole-linked 1,2,3-triazole congeners as agentsMethyl 3-[(6-nitro-4-oxo-3-phenyl-3,4-di-hydro-quinazolin-2-yl)sulfan-yl]propano-ateSynthesis, Biological Evaluation and Docking Analysis of Some Novel Quinazolin Derivatives as Antitumor Agents.Chemical characteristics, synthetic methods, and biological potential of quinazoline and quinazolinone derivatives.Synthesis and biological evaluation of 2-aminobenzamide derivatives as antimicrobial agents: opening/closing pharmacophore site.Synthesis, anticancer and apoptosis-inducing activities of quinazoline-isatin conjugates: epidermal growth factor receptor-tyrosine kinase assay and molecular docking studies.Biologically Active Heterocyclic Hybrids Based on Quinazolinone, Benzofuran and Imidazolium Moieties: Synthesis, Characterization, Cytotoxic and Antibacterial Evaluation.Synthesis and In Vitro Cytotoxic Properties of Polycarbo-Substituted 4-(Arylamino)quinazolines.Synthesis and cytotoxicity evaluation of some new 6-nitro derivatives of thiazole-containing 4-(3H)-quinazolinone.Reactivity of 2-ethoxyquinazolin- 4-yl hydrazine and its use in synthesis of novel quinazoline derivatives of antimicrobial activitySynthesis and Anticancer Activities of Novel Guanylhydrazone and Aminoguanidine Tetrahydropyran Derivatives.Synthesis and potential antitumor activity of 7-(4-substituted piperazin-1-yl)-4-oxoquinolines based on ciprofloxacin and norfloxacin scaffolds: in silico studies.Synthesis, antitumor and antimicrobial activity of some new 6-methyl-3-phenyl-4(3H)-quinazolinone analogues: in silico studies.Design, synthesis and in vitro antiproliferative activity of novel isatin-quinazoline hybrids.The safety and efficacy of vandetanib in the treatment of progressive medullary thyroid cancer.Design and synthesis of quinazolinone tagged acridones as cytotoxic agents and their effects on EGFR tyrosine kinase.Synthesis, antitumor evaluation and docking study of novel 4-anilinoquinazoline derivatives as potential epidermal growth factor receptor (EGFR) inhibitors.2-alkyl(aryl)-quinazolin-4(3H)-thiones, 2-R-(quinazolin-4(3H)-ylthio)carboxylic acids and amides: synthesis, molecular docking, antimicrobial and anticancer properties.Antibacterial, antifungal and cytotoxic evaluation of some new 2,3-disubstituted 4(3H)-quinazolinone derivatives.2-{[2-Methyl-3-(2-methyl-phen-yl)-4-oxo-3,4-dihydro-quinazolin-8-yl]-oxy}acetonitrile.2-Methyl-3-(2-methyl-phen-yl)-4-oxo-3,4-dihydro-quinazolin-8-yl 4-methyl-benzoate.2-Methyl-3-(2-methyl-phen-yl)-7-nitro-quinazolin-4(3H)-one.2-Methyl-3-(2-methyl-phen-yl)-4-oxo-3,4-dihydro-quinazolin-8-yl thio-phene-2-carboxyl-ate.2-Methyl-3-(2-methyl-phen-yl)-4-oxo-3,4-dihydro-quinazolin-8-yl 4-bromo-benzene-1-sulfonate.(S,E)-3-[(2-Hy-droxy-benzyl-idene)amino]-2-(2-hy-droxy-phen-yl)-2,3-dihydro-quinazolin-4(1H)-oneDocking study, synthesis and antimicrobial evaluation of some novel 4-anilinoquinazoline derivatives.8-Benz-yloxy-2-methyl-3-(2-methyl-phenyl)quinazolin-4(3H)-one.6-Methyl-3-phenyl-2-sulfanyl-idene-1,2,3,4-tetra-hydro-quinazolin-4-one.2-Methyl-3-(2-methyl-phen-yl)-4-oxo-3,4-dihydro-quinazolin-8-yl benzoate.Synthesis and anticancer activity of new quinazoline derivatives.Synthesis and characterization of quinazoline derivatives: search for hybrid molecule as diuretic and antihypertensive agents.Synthesis and biological evaluation of 2-styrylquinolines as antitumour agents and EGFR kinase inhibitors: molecular docking study.Synthesis, in vitro antitumour activity, and molecular docking study of novel 2-substituted mercapto-3-(3,4,5-trimethoxybenzyl)-4(3H)-quinazolinone analogues.Synthesis, antitumour and antioxidant activities of novel α,β-unsaturated ketones and related heterocyclic analogues: EGFR inhibition and molecular modelling study.
P2860
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P2860
Design, synthesis and biological evaluation of novel quinazoline derivatives as potential antitumor agents: molecular docking study.
description
2010 nî lūn-bûn
@nan
2010年の論文
@ja
2010年論文
@yue
2010年論文
@zh-hant
2010年論文
@zh-hk
2010年論文
@zh-mo
2010年論文
@zh-tw
2010年论文
@wuu
2010年论文
@zh
2010年论文
@zh-cn
name
Design, synthesis and biologic ...... ents: molecular docking study.
@en
Design, synthesis and biologic ...... ents: molecular docking study.
@nl
type
label
Design, synthesis and biologic ...... ents: molecular docking study.
@en
Design, synthesis and biologic ...... ents: molecular docking study.
@nl
prefLabel
Design, synthesis and biologic ...... ents: molecular docking study.
@en
Design, synthesis and biologic ...... ents: molecular docking study.
@nl
P2093
P50
P1476
Design, synthesis and biologic ...... gents: molecular docking study
@en
P2093
Abdulaziz M Aleisa
Alaa A-M Abdel-Aziz
Mohamed M Sayed-Ahmed
Naglaa I Abdel-Aziz
Sami G Abdel-Hamide
P304
P356
10.1016/J.EJMECH.2010.06.013
P577
2010-06-16T00:00:00Z