Identification of a Chemical Probe for Family VIII Bromodomains through Optimization of a Fragment Hit
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Targeting the Bromome: are we there yet?Chemical probes targeting epigenetic proteins: Applications beyond oncology.Discovery of a PCAF Bromodomain Chemical Probe.Bromodomains in Protozoan Parasites: Evolution, Function, and Opportunities for Drug Development.Mammalian SWI/SNF complexes in cancer: emerging therapeutic opportunities.Chemical modulators for epigenome reader domains as emerging epigenetic therapies for cancer and inflammation.Chemical probes and inhibitors of bromodomains outside the BET family.Crystal structure of (1S,4S)-2,5-diazo-niabi-cyclo[2.2.1]heptane dibromide.Temporal regulation of chromatin during myoblast differentiation.The BRG1 ATPase of human SWI/SNF chromatin remodeling enzymes as a driver of cancer.Large-scale analysis of water stability in bromodomain binding pockets with grand canonical Monte CarloDiscovery of a PCAF Bromodomain Chemical Probe
P2860
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P2860
Identification of a Chemical Probe for Family VIII Bromodomains through Optimization of a Fragment Hit
description
2016 nî lūn-bûn
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2016年の論文
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2016年学术文章
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2016年学术文章
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2016年学术文章
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2016年学术文章
@zh-my
2016年学术文章
@zh-sg
2016年學術文章
@yue
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2016年學術文章
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name
Identification of a Chemical P ...... Optimization of a Fragment Hit
@en
Identification of a Chemical P ...... ptimization of a Fragment Hit.
@nl
type
label
Identification of a Chemical P ...... Optimization of a Fragment Hit
@en
Identification of a Chemical P ...... ptimization of a Fragment Hit.
@nl
prefLabel
Identification of a Chemical P ...... Optimization of a Fragment Hit
@en
Identification of a Chemical P ...... ptimization of a Fragment Hit.
@nl
P2093
P2860
P50
P1476
Identification of a Chemical P ...... Optimization of a Fragment Hit
@en
P2093
Adam D Torrey
Alexandria Taylor
Alison O'Mahony
Anthony N Imbalzano
Brian S Gerstenberger
Brian Samas
Brian T Nasipak
Catherine Rogers
Cynthia Tallant
Dafydd R Owen
P2860
P304
P356
10.1021/ACS.JMEDCHEM.6B00012
P407
P50
P577
2016-04-26T00:00:00Z