Brain access and anticonvulsant efficacy of carbamazepine, lamotrigine, and felbamate in ABCC2/MRP2-deficient TR- rats.
about
Targeting multidrug resistance in cancerBlood-brain barrier active efflux transporters: ATP-binding cassette gene family.Drug resistance in epilepsy: putative neurobiologic and clinical mechanisms.Structure and function of the MRP2 (ABCC2) protein and its role in drug disposition.The emerging importance of transporter proteins in the psychopharmacological treatment of the pregnant patient.Recent advances in 2D and 3D in vitro systems using primary hepatocytes, alternative hepatocyte sources and non-parenchymal liver cells and their use in investigating mechanisms of hepatotoxicity, cell signaling and ADME.One of the hottest topics in epileptology: ABC proteins. Their inhibition may be the future for patients with intractable seizures.Genetic Variations of ABCC2 Gene Associated with Adverse Drug Reactions to Valproic Acid in Korean Epileptic PatientsPrediction of antiepileptic drug efficacy: the use of intracerebral microdialysis to monitor biophase concentrations.New insights in the biology of ABC transporters ABCC2 and ABCC3: impact on drug disposition.Exploring the Carbamazepine Interaction with Human Pregnane X Receptor and Effect on ABCC2 Using in Vitro and in Silico Approach.Neural overexpression of multidrug resistance-associated protein 1 and refractory epilepsy: a meta-analysis of nine studies.ABCC2 polymorphisms and haplotype are associated with drug resistance in Chinese epileptic patients.A pilot study on brain-to-plasma partition of 10,11-dyhydro-10-hydroxy-5H-dibenzo(b,f)azepine-5-carboxamide and MDR1 brain expression in epilepsy patients not responding to oxcarbazepine.Lack of interactions between breast cancer resistance protein (bcrp/abcg2) and selected antiepileptic agents.Upregulation of brain expression of P-glycoprotein in MRP2-deficient TR(-) rats resembles seizure-induced up-regulation of this drug efflux transporter in normal rats.
P2860
Q29616803-83F00F7B-75F2-45D9-B484-CC0FFA2E83B9Q33985133-863D5A85-CA90-4EB8-9ED6-EE43160D1E4EQ36157234-B76AC220-1CFA-45BF-B7B6-8A52576772BCQ36544905-4CCEB079-B5DA-472A-BDEB-28EA03537410Q37024001-B2AA3DB9-FC57-40FB-836F-D8A8C968C896Q37121662-C01FF509-89CD-4FF0-93EB-39695081C068Q37204397-1C57FF16-D7C2-4F41-80FB-630627342DD8Q37500912-FA6A251F-0119-44AF-B019-B38DE390BF86Q37554396-0BD01748-473F-4A2A-956F-1B4873CC09F5Q38266172-B2F11EF9-D2CC-4FC6-8E3D-E0E8D33BD29AQ38706504-E8625F81-B8B6-4B0C-89E4-937FEF036273Q40911740-63B7D93A-228F-4CB1-A373-FFF2E7AAE830Q43903895-C9855DA4-14D2-4CC3-AE04-8BAF549CD5C5Q46725875-39C4BC50-EA82-4435-9CB0-CDF11DA2A7ADQ46984881-C4D322D0-A22F-40C1-BCFC-F423BC369D72Q48201303-ECDE828F-E5C7-4707-B751-6A39E06A8F57
P2860
Brain access and anticonvulsant efficacy of carbamazepine, lamotrigine, and felbamate in ABCC2/MRP2-deficient TR- rats.
description
2003 nî lūn-bûn
@nan
2003年の論文
@ja
2003年論文
@yue
2003年論文
@zh-hant
2003年論文
@zh-hk
2003年論文
@zh-mo
2003年論文
@zh-tw
2003年论文
@wuu
2003年论文
@zh
2003年论文
@zh-cn
name
Brain access and anticonvulsan ...... ABCC2/MRP2-deficient TR- rats.
@en
type
label
Brain access and anticonvulsan ...... ABCC2/MRP2-deficient TR- rats.
@en
prefLabel
Brain access and anticonvulsan ...... ABCC2/MRP2-deficient TR- rats.
@en
P2860
P1433
P1476
Brain access and anticonvulsan ...... ABCC2/MRP2-deficient TR- rats.
@en
P2093
Maren Fedrowitz
Wolfgang Löscher
P2860
P304
P356
10.1111/J.0013-9580.2003.22603.X
P577
2003-12-01T00:00:00Z