Coupling of the human A1 adenosine receptor to different heterotrimeric G proteins: evidence for agonist-specific G protein activation.
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Antagonist affinity measurements at the Gi-coupled human histamine H3 receptor expressed in CHO cellsAdenosine A(1) receptor agonist N(6)-cyclohexyl-adenosine induced phosphorylation of delta opioid receptor and desensitization of its signaling.Effect of adenosine on membrane potential and Ca2+ in juxtaglomerular cells. Comparison with angiotensin IIThe cannabinoid agonist WIN55,212-2 increases intracellular calcium via CB1 receptor coupling to Gq/11 G proteins.Structural determinants in the second intracellular loop of the human cannabinoid CB1 receptor mediate selective coupling to G(s) and G(i)Purinergic system dysfunction in mood disorders: a key target for developing improved therapeutics.Noradrenaline stimulates cell proliferation by suppressing potassium channels via G(i/o) -protein-coupled α(1B) -adrenoceptors in human osteoblasts.On the selectivity of the Gαq inhibitor UBO-QIC: A comparison with the Gαi inhibitor pertussis toxin.Allosteric modulation and functional selectivity of G protein-coupled receptors.Multiple GPCR conformations and signalling pathways: implications for antagonist affinity estimates.Tissue-nonspecific alkaline phosphatase acts redundantly with PAP and NT5E to generate adenosine in the dorsal spinal cord.Internalization and desensitization of adenosine receptors.Stereochemistry of an agonist determines coupling preference of beta2-adrenoceptor to different G proteins in cardiomyocytesQuantification of Gi-mediated inhibition of adenylyl cyclase activity reveals that UDP is a potent agonist of the human P2Y14 receptor.Functional selectivity of adenosine receptor ligandsFunctional signaling biases in G protein-coupled receptors: Game Theory and receptor dynamics.Allosteric interactions at adenosine A(1) and A(3) receptors: new insights into the role of small molecules and receptor dimerization.Purinergic Receptor Expression and Potential Association with Human Embryonic Stem Cell-Derived Oligodendrocyte Progenitor Cell Development.Extracellular cAMP activates molecular signalling pathways associated with sperm capacitation in bovines.A1 Adenosine Receptor Activation Modulates Central Nervous System Development and Repair.Influence of fluorophore and linker composition on the pharmacology of fluorescent adenosine A1 receptor ligands.Modulation of adenosine A1 and A2A receptors in C6 glioma cells during hypoxia: involvement of endogenous adenosine.GPR93 activation by protein hydrolysate induces CCK transcription and secretion in STC-1 cells.Different response patterns of several ligands at the sphingosine-1-phosphate receptor subtype 3 (S1P(3))Plasticity within striatal direct pathway neurons after neonatal dopamine depletion is mediated through a novel functional coupling of serotonin 5-HT2 receptors to the ERK 1/2 map kinase pathway.Co-localization and functional cross-talk between A1 and P2Y1 purine receptors in rat hippocampus.Modelling and simulation of biased agonism dynamics at a G protein-coupled receptor.Calcium receptor signaling and citrate transport.4-amino-6-alkyloxy-2-alkylthiopyrimidine derivatives as novel non-nucleoside agonists for the adenosine A1 receptor.
P2860
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P2860
Coupling of the human A1 adenosine receptor to different heterotrimeric G proteins: evidence for agonist-specific G protein activation.
description
2004 nî lūn-bûn
@nan
2004年の論文
@ja
2004年論文
@yue
2004年論文
@zh-hant
2004年論文
@zh-hk
2004年論文
@zh-mo
2004年論文
@zh-tw
2004年论文
@wuu
2004年论文
@zh
2004年论文
@zh-cn
name
Coupling of the human A1 adeno ...... specific G protein activation.
@en
Coupling of the human A1 adeno ...... specific G protein activation.
@nl
type
label
Coupling of the human A1 adeno ...... specific G protein activation.
@en
Coupling of the human A1 adeno ...... specific G protein activation.
@nl
prefLabel
Coupling of the human A1 adeno ...... specific G protein activation.
@en
Coupling of the human A1 adeno ...... specific G protein activation.
@nl
P2860
P356
P1476
Coupling of the human A1 adeno ...... specific G protein activation.
@en
P2093
Yolande Cordeaux
P2860
P304
P356
10.1038/SJ.BJP.0705925
P407
P577
2004-08-09T00:00:00Z