Structure-activity relationship, biological, and pharmacological characterization of the proline sulfonamide ACT-462206: a potent, brain-penetrant dual orexin 1/orexin 2 receptor antagonist.
about
Orexin receptor antagonists--a patent review (2010 to August 2014).Orexin OX2 Receptor Antagonists as Sleep Aids.Substituted cyclopentanes, tetrahydrofurans and pyrrolidines as orexin-1-receptor antagonists for treatment of various CNS disorders (WO2015/055994; WO2015/124932; WO2015/124934).Orexin research: patent news from 2016.Discovery of Highly Potent Dual Orexin Receptor Antagonists via a Scaffold-Hopping Approach.Orexin Receptor Antagonists
P2860
Structure-activity relationship, biological, and pharmacological characterization of the proline sulfonamide ACT-462206: a potent, brain-penetrant dual orexin 1/orexin 2 receptor antagonist.
description
2014 nî lūn-bûn
@nan
2014年の論文
@ja
2014年論文
@yue
2014年論文
@zh-hant
2014年論文
@zh-hk
2014年論文
@zh-mo
2014年論文
@zh-tw
2014年论文
@wuu
2014年论文
@zh
2014年论文
@zh-cn
name
Structure-activity relationshi ...... /orexin 2 receptor antagonist.
@en
Structure-activity relationshi ...... /orexin 2 receptor antagonist.
@nl
type
label
Structure-activity relationshi ...... /orexin 2 receptor antagonist.
@en
Structure-activity relationshi ...... /orexin 2 receptor antagonist.
@nl
prefLabel
Structure-activity relationshi ...... /orexin 2 receptor antagonist.
@en
Structure-activity relationshi ...... /orexin 2 receptor antagonist.
@nl
P2093
P2860
P356
P1433
P1476
Structure-activity relationshi ...... /orexin 2 receptor antagonist.
@en
P2093
Alexander Treiber
Bibia Heidmann
Catherine Roch-Brisbare
Christine Brotschi
Christoph Boss
Francois Jenck
Hamed Aissaoui
Hendrik Dietrich
Jodi T Williams
John Gatfield
P2860
P304
P356
10.1002/CMDC.201402258
P577
2014-08-21T00:00:00Z