Ring substituted and other conformationally constrained tyrosine analogues of [D-Pen2,D-Pen5]enkephalin with delta opioid receptor selectivity.

Ring substituted and other conformationally constrained tyrosine analogues of [D-Pen2,D-Pen5]enkephalin with delta opioid receptor selectivity.

Item
http://www.wikidata.org/entity/Q44331217
A three-dimensional model of the delta-opioid pharmacophore: comparative molecular modeling of peptide and nonpeptide ligands.Biological and conformational evaluation of bifunctional compounds for opioid receptor agonists and neurokinin 1 receptor antagonists possessing two penicillaminesImproving metabolic stability by glycosylation: bifunctional peptide derivatives that are opioid receptor agonists and neurokinin 1 receptor antagonistsThe biological activity and metabolic stability of peptidic bifunctional compounds that are opioid receptor agonists and neurokinin-1 receptor antagonists with a cystine moiety.Conformationally constrained histidines in the design of peptidomimetics: strategies for the χ-space control.Assessment of stereoselectivity of trimethylphenylalanine analogues of delta-opioid [D-Pen(2),D-Pen(5)]-enkephalin.Chemoselective nitration of phenols with tert-butyl nitrite in solution and on solid support.Synthesis of stable and potent delta/mu opioid peptides: analogues of H-Tyr-c[D-Cys-Gly-Phe-D-Cys]-OH by ring-closing metathesis.Dynorphin A analogs containing a conformationally constrained phenylalanine derivative in position 4: reversal of preferred stereochemistry for opioid receptor affinity and discrimination of kappa vs. delta receptors.Conformational restriction of Tyr and Phe side chains in opioid peptides: information about preferred and bioactive side-chain topology.Analysis of N-amino-imidazolin-2-one peptide turn mimic 4-position substituent effects on conformation by X-ray crystallography.Design of peptides, proteins, and peptidomimetics in chi space.
P2860

Ring substituted and other conformationally constrained tyrosine analogues of [D-Pen2,D-Pen5]enkephalin with delta opioid receptor selectivity.

Item
http://www.wikidata.org/entity/Q44331217
description
1992 nî lūn-bûn
@nan
1992年の論文
@ja
1992年学术文章
@wuu
1992年学术文章
@zh
1992年学术文章
@zh-cn
1992年学术文章
@zh-hans
1992年学术文章
@zh-my
1992年学术文章
@zh-sg
1992年學術文章
@yue
1992年學術文章
@zh-hant
name
Ring substituted and other con ...... a opioid receptor selectivity.
@en
Ring substituted and other con ...... a opioid receptor selectivity.
@nl
type
label
Ring substituted and other con ...... a opioid receptor selectivity.
@en
Ring substituted and other con ...... a opioid receptor selectivity.
@nl
prefLabel
Ring substituted and other con ...... a opioid receptor selectivity.
@en
Ring substituted and other con ...... a opioid receptor selectivity.
@nl
P1433
P1476
P2093
P304
P31
P356
P407
P433
P478
P577
P698
P921
P356
P1433
P1476
Ring substituted and other con ...... a opioid receptor selectivity.
@en
P2093
P304
P31
P356
P407
P433
P478
P577
P698
P921