Optimization of a "bump-and-hole" approach to allele-selective BET bromodomain inhibition.

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Optimization of a "bump-and-hole" approach to allele-selective BET bromodomain inhibition.

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2018 nî lūn-bûn

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2018年の論文

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2018年学术文章

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Optimization of a "bump-and-ho ...... ve BET bromodomain inhibition.

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Optimization of a "bump-and-ho ...... ve BET bromodomain inhibition.

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Optimization of a "bump-and-ho ...... ve BET bromodomain inhibition.

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Optimization of a "bump-and-ho ...... ve BET bromodomain inhibition.

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Optimization of a "bump-and-ho ...... ve BET bromodomain inhibition.

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Optimization of a "bump-and-ho ...... ve BET bromodomain inhibition.

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P1476

Optimization of a "bump-and-ho ...... ve BET bromodomain inhibition.

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P2093

A Brien

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A Testa

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K D Read

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L C J Ellis

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L van Beurden

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M Zengerle

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O Epemolu

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V Coulthard

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P2860

Brd4 maintains constitutively active NF-κB in cancer cells by binding to acetylated RelA

Selective inhibition of BET bromodomains

Brd4 coactivates transcriptional activation of NF-kappaB via specific binding to acetylated RelA

Histone recognition and large-scale structural analysis of the human bromodomain family

Disrupting the interaction of BRD4 with diacetylated Twist suppresses tumorigenesis in basal-like breast cancer

Chemical genetics approaches for selective intervention in epigenetics

Suppression of inflammation by a synthetic histone mimic

Inhibition of BET recruitment to chromatin as an effective treatment for MLL-fusion leukaemia

RVX-208, an inhibitor of BET transcriptional regulators with selectivity for the second bromodomain

Selective Chemical Modulation of Gene Transcription Favors Oligodendrocyte Lineage Progression

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2452-2468

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scholarly article

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10.1039/C7SC02536J

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P433

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P478

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2018-01-24T00:00:00Z

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29732121

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5909127

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