about
Drug discovery: Designing the ideal opioidMembrane potentials regulating GPCRs: insights from experiments and molecular dynamics simulationsCentral mediators involved in the febrile response: effects of antipyretic drugsFluorescent approaches for understanding interactions of ligands with G protein coupled receptorsThe photochemical determinants of color vision: revealing how opsins tune their chromophore's absorption wavelengthSerial Femtosecond Crystallography of G Protein-Coupled ReceptorsMolecular control of δ-opioid receptor signallingStructure of the human P2Y12 receptor in complex with an antithrombotic drugStructural insights into ligand recognition and selectivity for classes A, B, and C GPCRsTransmembrane recognition of the semaphorin co-receptors neuropilin 1 and plexin A1: coarse-grained simulationsTSH Receptor Signaling Abrogation by a Novel Small MoleculeInvited review: GPCR structural characterization: Using fragments as building blocks to determine a complete structure.The role of experimental and computational structural approaches in 7TM drug discovery.Structural-Functional Features of the Thyrotropin Receptor: A Class A G-Protein-Coupled Receptor at WorkG protein-coupled receptors in cardiac biology: old and new receptorsDifferences in allosteric communication pipelines in the inactive and active states of a GPCR.Allosteric sodium in class A GPCR signalingPlatelets and cancer: a casual or causal relationship: revisited.Conserved Residues Control Activation of Mammalian G Protein-Coupled Odorant Receptors.The Importance of Ligand-Receptor Conformational Pairs in Stabilization: Spotlight on the N/OFQ G Protein-Coupled ReceptorAllosteric signaling through an mGlu2 and 5-HT2A heteromeric receptor complex and its potential contribution to schizophreniaIndividual variation of human S1P₁ coding sequence leads to heterogeneity in receptor function and drug interactionsIn silico study on binding specificity of gonadotropins and their receptors: design of a novel and selective peptidomimetic for human follicle stimulating hormone receptor.New small molecule agonists to the thyrotropin receptor.In vivo properties of KNT-127, a novel δ opioid receptor agonist: receptor internalization, antihyperalgesia and antidepressant effects in mice.Why we need many more G protein-coupled receptor structuresThe role of membrane curvature elastic stress for function of rhodopsin-like G protein-coupled receptorsEpigenetic dysregulation of hairy and enhancer of split 4 (HES4) is associated with striatal degeneration in postmortem Huntington brains.A pepducin derived from the third intracellular loop of FPR2 is a partial agonist for direct activation of this receptor in neutrophils but a full agonist for cross-talk triggered reactivation of FPR2.Quantitative Measurement of GPCR Endocytosis via Pulse-Chase Covalent Labeling.Monitoring β-arrestin recruitment via β-lactamase enzyme fragment complementation: purification of peptide E as a low-affinity ligand for mammalian bombesin receptors.Targeting the thyroid-stimulating hormone receptor with small molecule ligands and antibodiesComparative analyses of downstream signal transduction targets modulated after activation of the AT1 receptor by two β-arrestin-biased agonists.Allosteric Activation of a G Protein-coupled Receptor with Cell-penetrating Receptor MimeticsInsights into Basal Signaling Regulation, Oligomerization, and Structural Organization of the Human G-Protein Coupled Receptor 83.Elucidation of molecular kinetic schemes from macroscopic traces using system identification.Optimising the combination of thermostabilising mutations in the neurotensin receptor for structure determination.Acting on Hormone Receptors with Minimal Side Effect on Cell Proliferation: A Timely Challenge Illustrated with GLP-1R and GPERSupra-physiological efficacy at GPCRs: superstition or super agonists?Computational Prediction and Biochemical Analyses of New Inverse Agonists for the CB1 Receptor
P2860
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P2860
description
2012 nî lūn-bûn
@nan
2012 թուականի Սեպտեմբերին հրատարակուած գիտական յօդուած
@hyw
2012 թվականի սեպտեմբերին հրատարակված գիտական հոդված
@hy
2012年の論文
@ja
2012年論文
@yue
2012年論文
@zh-hant
2012年論文
@zh-hk
2012年論文
@zh-mo
2012年論文
@zh-tw
2012年论文
@wuu
name
Restructuring G-protein- coupled receptor activation
@ast
Restructuring G-protein- coupled receptor activation
@en
Restructuring G-protein- coupled receptor activation
@nl
type
label
Restructuring G-protein- coupled receptor activation
@ast
Restructuring G-protein- coupled receptor activation
@en
Restructuring G-protein- coupled receptor activation
@nl
prefLabel
Restructuring G-protein- coupled receptor activation
@ast
Restructuring G-protein- coupled receptor activation
@en
Restructuring G-protein- coupled receptor activation
@nl
P3181
P1433
P1476
Restructuring G-protein- coupled receptor activation
@en
P2093
Martin Audet
P3181
P356
10.1016/J.CELL.2012.09.003
P407
P577
2012-09-28T00:00:00Z