An antifungal agent inhibits an aminoacyl-tRNA synthetase by trapping tRNA in the editing site
about
Topical and device-based treatments for fungal infections of the toenailsNew agents for the treatment of drug-resistant Mycobacterium tuberculosisThe tRNA Elbow in Structure, Recognition and EvolutionSpotlight on tavaborole for the treatment of onychomycosisEvolutionary Limitation and Opportunities for Developing tRNA Synthetase Inhibitors with 5-Binding-Mode ClassificationtRNAs as antibiotic targetsMetalloid compounds as drugsIn silico discovery of aminoacyl-tRNA synthetase inhibitorsDiscovery of Novel Oral Protein Synthesis Inhibitors of Mycobacterium tuberculosis That Target Leucyl-tRNA SynthetaseBoron Mimetics: 1,2-Dihydro-1,2-azaborines Bind inside a Nonpolar Cavity of T4 LysozymeCrystal structures of Saccharomyces cerevisiae tryptophanyl-tRNA synthetase: new insights into the mechanism of tryptophan activation and implications for anti-fungal drug designPeripheral insertion modulates the editing activity of the isolated CP1 domain of leucyl-tRNA synthetaseATP-directed capture of bioactive herbal-based medicine on human tRNA synthetaseDiscovery of a Novel Class of Boron-Based Antibacterials with Activity against Gram-Negative BacteriaCrystal structures of Plasmodium falciparum cytosolic tryptophanyl-tRNA synthetase and its potential as a target for structure-guided drug designCo-crystal structure of a T-box riboswitch stem I domain in complex with its cognate tRNADiscovery of a potent benzoxaborole-based anti-pneumococcal agent targeting leucyl-tRNA synthetaseStructural dynamics of the aminoacylation and proofreading functional cycle of bacterial leucyl-tRNA synthetasePlant tumour biocontrol agent employs a tRNA-dependent mechanism to inhibit leucyl-tRNA synthetaseThe physiological target for LeuRS translational quality control is norvalineStructural analysis of malaria-parasite lysyl-tRNA synthetase provides a platform for drug developmentBenzoxaborole as a new chemotype for carbonic anhydrase inhibitionAnalogs of natural aminoacyl-tRNA synthetase inhibitors clear malaria in vivoA genomic glimpse of aminoacyl-tRNA synthetases in malaria parasite Plasmodium falciparumApplication of Nail Polish During Topical Management of Onychomycosis: Are Data Available to Guide the Clinician About What to Tell Their Patients?Genomic and Proteomic Studies on the Mode of Action of Oxaboroles against the African TrypanosomeProtein Translation Enzyme lysyl-tRNA Synthetase Presents a New Target for Drug Development against Causative Agents of Loiasis and SchistosomiasisComparative chemical genomics reveal that the spiroindolone antimalarial KAE609 (Cipargamin) is a P-type ATPase inhibitorA potent antimalarial benzoxaborole targets a Plasmodium falciparum cleavage and polyadenylation specificity factor homologueStructural basis for full-spectrum inhibition of translational functions on a tRNA synthetaseDiscovery of novel benzoxaborole-based potent antitrypanosomal agents.tRNA-dependent pre-transfer editing by prokaryotic leucyl-tRNA synthetase.Ligand co-crystallization of aminoacyl-tRNA synthetases from infectious disease organismstRNA synthetase: tRNA aminoacylation and beyondThe balance between pre- and post-transfer editing in tRNA synthetases.A paradigm shift for the amino acid editing mechanism of human cytoplasmic leucyl-tRNA synthetase.Functional segregation of a predicted "hinge" site within the beta-strand linkers of Escherichia coli leucyl-tRNA synthetasePartitioning of tRNA-dependent editing between pre- and post-transfer pathways in class I aminoacyl-tRNA synthetases.Discovery of novel orally bioavailable oxaborole 6-carboxamides that demonstrate cure in a murine model of late-stage central nervous system african trypanosomiasis.Antibiotics and bacterial resistance in the 21st century.
P2860
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P2860
An antifungal agent inhibits an aminoacyl-tRNA synthetase by trapping tRNA in the editing site
description
2007 nî lūn-bûn
@nan
2007 թուականի Յունիսին հրատարակուած գիտական յօդուած
@hyw
2007 թվականի հունիսին հրատարակված գիտական հոդված
@hy
2007年の論文
@ja
2007年論文
@yue
2007年論文
@zh-hant
2007年論文
@zh-hk
2007年論文
@zh-mo
2007年論文
@zh-tw
2007年论文
@wuu
name
An antifungal agent inhibits a ...... pping tRNA in the editing site
@ast
An antifungal agent inhibits a ...... pping tRNA in the editing site
@en
An antifungal agent inhibits a ...... pping tRNA in the editing site
@nl
type
label
An antifungal agent inhibits a ...... pping tRNA in the editing site
@ast
An antifungal agent inhibits a ...... pping tRNA in the editing site
@en
An antifungal agent inhibits a ...... pping tRNA in the editing site
@nl
prefLabel
An antifungal agent inhibits a ...... pping tRNA in the editing site
@ast
An antifungal agent inhibits a ...... pping tRNA in the editing site
@en
An antifungal agent inhibits a ...... pping tRNA in the editing site
@nl
P2093
P2860
P3181
P356
P1433
P1476
An antifungal agent inhibits a ...... pping tRNA in the editing site
@en
P2093
Anya Yaremchuk
Fernando L Rock
Huchen Zhou
Jacob J Plattner
Lucy Shapiro
M R K Alley
Mikhail Tukalo
Stephen J Baker
Stephen J Benkovic
Susan A Martinis
P2860
P304
P3181
P356
10.1126/SCIENCE.1142189
P407
P577
2007-06-22T00:00:00Z