Selective and brain-permeable polo-like kinase-2 (Plk-2) inhibitors that reduce α-synuclein phosphorylation in rat brain
about
Small molecule annotation for the Protein Data Bank.Modelling Ser129 phosphorylation inhibits membrane binding of pore-forming alpha-synuclein oligomersCurrent progress and future perspectives in the development of anti-polo-like kinase 1 therapeutic agents.Discovery of 2-(1H-indol-5-ylamino)-6-(2,4-difluorophenylsulfonyl)-8-methylpyrido[2,3-d]pyrimidin-7(8H)-one (7ao) as a potent selective inhibitor of Polo like kinase 2 (PLK2).Polo-like kinase 2 acting as a promoter in human tumor cells with an abundance of TAp73.Recent Advances and New Strategies in Targeting Plk1 for Anticancer TherapyPLK2 phosphorylates and inhibits enriched TAp73 in human osteosarcoma cellsAge- and brain region-dependent α-synuclein oligomerization is attributed to alterations in intrinsic enzymes regulating α-synuclein phosphorylation in aging monkey brains.Highly Atom Economic Synthesis of d-2-Aminobutyric Acid through an In Vitro Tri-enzymatic Catalytic SystemPlk2 Loss Commonly Occurs in Colorectal Carcinomas but not Adenomas: Relationship to mTOR Signaling.
P2860
Q30872013-1F511EDF-057D-4BC5-80B1-BEABA626ABD7Q31165000-A6FA37C6-F3C5-40CF-BC3B-1E0527AE90C0Q33873351-124DB1FB-EBF2-4ABC-B9AF-3F60D25FA0A0Q35893205-101DF330-6699-4C61-ACDF-B3B00FD61C69Q36326031-28DDEAC2-1223-47C1-B218-736E8AA42E5BQ36386336-44AD9370-34C3-4677-9232-774AB2432900Q36451518-2FCD4E3F-5E72-4852-9F94-AE4BCDAC8F10Q36962314-C2C64D8B-039E-4847-B11B-DB716EDD08C3Q41239574-A43804FF-397A-412C-82A5-B1E675D6B26EQ49968483-F3D07DC9-CEAD-4178-889A-BF22C918EE23
P2860
Selective and brain-permeable polo-like kinase-2 (Plk-2) inhibitors that reduce α-synuclein phosphorylation in rat brain
description
2013 nî lūn-bûn
@nan
2013 թուականի Օգոստոսին հրատարակուած գիտական յօդուած
@hyw
2013 թվականի օգոստոսին հրատարակված գիտական հոդված
@hy
2013年の論文
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2013年論文
@yue
2013年論文
@zh-hant
2013年論文
@zh-hk
2013年論文
@zh-mo
2013年論文
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2013年论文
@wuu
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Selective and brain-permeable ...... n phosphorylation in rat brain
@ast
Selective and brain-permeable ...... n phosphorylation in rat brain
@en
Selective and brain-permeable ...... n phosphorylation in rat brain
@nl
type
label
Selective and brain-permeable ...... n phosphorylation in rat brain
@ast
Selective and brain-permeable ...... n phosphorylation in rat brain
@en
Selective and brain-permeable ...... n phosphorylation in rat brain
@nl
prefLabel
Selective and brain-permeable ...... n phosphorylation in rat brain
@ast
Selective and brain-permeable ...... n phosphorylation in rat brain
@en
Selective and brain-permeable ...... n phosphorylation in rat brain
@nl
P2093
P2860
P921
P356
P1433
P1476
Selective and brain-permeable ...... n phosphorylation in rat brain
@en
P2093
Andrei W Konradi
Anh P Truong
Danielle L Aubele
Dean R Artis
Donald Fauss
George Tonn
Heather Zhang
Hing L Sham
P2860
P304
P356
10.1002/CMDC.201300166
P577
2013-08-01T00:00:00Z