Novel phenolic inhibitors of small/intermediate-conductance Ca²⁺-activated K⁺ channels, KCa3.1 and KCa2.3
about
Pharmacological gating modulation of small- and intermediate-conductance Ca(2+)-activated K(+) channels (KCa2.x and KCa3.1)A novel pan-negative-gating modulator of KCa2/3 channels, fluoro-di-benzoate, RA-2, inhibits endothelium-derived hyperpolarization-type relaxation in coronary artery and produces bradycardia in vivo.High expression of KCa3.1 in patients with clear cell renal carcinoma predicts high metastatic risk and poor survival.Modulation of K(Ca)3.1 channels by eicosanoids, omega-3 fatty acids, and molecular determinantsTungstate-targeting of BKαβ1 channels tunes ERK phosphorylation and cell proliferation in human vascular smooth muscle.Genetic deficit of KCa 3.1 channels protects against pulmonary circulatory collapse induced by TRPV4 channel activation.Inhibition of Intermediate-Conductance Calcium-Activated K Channel (KCa3.1) and Fibroblast Mitogenesis by α-Linolenic Acid and Alterations of Channel Expression in the Lysosomal Storage Disorders, Fabry Disease, and Niemann Pick CNuclear localization of the CK2α-subunit correlates with poor prognosis in clear cell renal cell carcinoma.Vascular Reactivity Profile of Novel KCa 3.1-Selective Positive-Gating Modulators in the Coronary Vascular Bed.Structural insights into the potency of SK channel positive modulators.Pharmacological activation of TRPV4 produces immediate cell damage and induction of apoptosis in human melanoma cells and HaCaT keratinocytes.9-Phenanthrol modulates postinhibitory rebound and afterhyperpolarizing potentials in an excitatory motor neuron of the medicinal leech.Rock Tea extract (Jasonia glutinosa) relaxes rat aortic smooth muscle by inhibition of L-type Ca(2+) channels.
P2860
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P2860
Novel phenolic inhibitors of small/intermediate-conductance Ca²⁺-activated K⁺ channels, KCa3.1 and KCa2.3
description
2013 nî lūn-bûn
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2013 թուականին հրատարակուած գիտական յօդուած
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2013 թվականին հրատարակված գիտական հոդված
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2013年の論文
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2013年論文
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2013年論文
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2013年論文
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2013年論文
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2013年論文
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2013年论文
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name
Novel phenolic inhibitors of s ...... K⁺ channels, KCa3.1 and KCa2.3
@ast
Novel phenolic inhibitors of s ...... K⁺ channels, KCa3.1 and KCa2.3
@en
Novel phenolic inhibitors of s ...... K⁺ channels, KCa3.1 and KCa2.3
@nl
type
label
Novel phenolic inhibitors of s ...... K⁺ channels, KCa3.1 and KCa2.3
@ast
Novel phenolic inhibitors of s ...... K⁺ channels, KCa3.1 and KCa2.3
@en
Novel phenolic inhibitors of s ...... K⁺ channels, KCa3.1 and KCa2.3
@nl
prefLabel
Novel phenolic inhibitors of s ...... K⁺ channels, KCa3.1 and KCa2.3
@ast
Novel phenolic inhibitors of s ...... K⁺ channels, KCa3.1 and KCa2.3
@en
Novel phenolic inhibitors of s ...... K⁺ channels, KCa3.1 and KCa2.3
@nl
P2860
P50
P1433
P1476
Novel phenolic inhibitors of s ...... ⁺ channels, KCa3.1 and KCa2.3.
@en
P2093
Heike Wulff
Ralf Köhler
P2860
P304
P356
10.1371/JOURNAL.PONE.0058614
P407
P50
P577
2013-03-14T00:00:00Z