about
Cardiac cAMP: production, hydrolysis, modulation and detectionRegulation of nephron water and electrolyte transport by adenylyl cyclasesSimilarly potent inhibition of adenylyl cyclase by P-site inhibitors in hearts from wild type and AC5 knockout miceA high throughput screening assay system for the identification of small molecule inhibitors of gspThe Concise Guide to PHARMACOLOGY 2013/14: enzymes.Prenatal programming of pulmonary hypertension induced by chronic hypoxia or ductal ligation in sheepcAMP-stimulated Cl- secretion is increased by glucocorticoids and inhibited by bumetanide in semicircular canal duct epithelium.Dissociations in the effects of β2-adrenergic receptor agonists on cAMP formation and superoxide production in human neutrophils: support for the concept of functional selectivity.Nucleotidyl cyclase activity of particulate guanylyl cyclase A: comparison with particulate guanylyl cyclases E and F, soluble guanylyl cyclase and bacterial adenylyl cyclases CyaA and edema factorIsoform selectivity of adenylyl cyclase inhibitors: characterization of known and novel compoundsDevelopment of a high-throughput screening paradigm for the discovery of small-molecule modulators of adenylyl cyclase: identification of an adenylyl cyclase 2 inhibitor.Generation and characterization of ATP analog-specific protein kinase Cδ.The adenylyl cyclase inhibitor MDL-12,330A potentiates insulin secretion via blockade of voltage-dependent K(+) channels in pancreatic beta cellsGuanylyl cyclases A and B are asymmetric dimers that are allosterically activated by ATP binding to the catalytic domain.Cyclic Adenosine 3',5'-Monophosphate Elevation and Biological Signaling through a Secretin Family Gs-Coupled G Protein-Coupled Receptor Are Restricted to a Single Adenylate Cyclase Isoform.Comparative electrostatic analysis of adenylyl cyclase for isoform dependent regulation properties.Identification of a selective small-molecule inhibitor of type 1 adenylyl cyclase activity with analgesic properties.Calmodulin-sensitive adenylyl cyclases mediate AVP-dependent cAMP production and Cl- secretion by human autosomal dominant polycystic kidney cells.A new site and mechanism of action for the widely used adenylate cyclase inhibitor SQ22,536Bithionol Potently Inhibits Human Soluble Adenylyl Cyclase through Binding to the Allosteric Activator SitePharmacological distinction between soluble and transmembrane adenylyl cyclases.Interactions of Bordetella pertussis adenylyl cyclase toxin CyaA with calmodulin mutants and calmodulin antagonists: comparison with membranous adenylyl cyclase I.Allosteric regulation of nucleotidyl cyclases: an emerging pharmacological target.Selectivity of pharmacological tools: implications for use in cell physiology. A review in the theme: Cell signaling: proteins, pathways and mechanisms.Adenosine receptors regulate gap junction coupling of the human cerebral microvascular endothelial cells hCMEC/D3 by Ca2+ influx through cyclic nucleotide-gated channels.International Union of Basic and Clinical Pharmacology. CI. Structures and Small Molecule Modulators of Mammalian Adenylyl Cyclases.Impairment of adenylyl cyclase 2 function and expression in hypoxanthine phosphoribosyltransferase-deficient rat B103 neuroblastoma cells as model for Lesch-Nyhan disease: BODIPY-forskolin as pharmacological tool.Epstein-Barr Virus-induced Gene 2 Mediates Allergen-induced Leukocyte Migration into Airways.Prostaglandin E2 Inhibits Histamine-Evoked Ca2+ Release in Human Aortic Smooth Muscle Cells through Hyperactive cAMP Signalling Junctions and Protein Kinase A.MDL-12330A potentiates TRAIL-induced apoptosis in gastric cancer cells through CHOP-mediated DR5 upregulation.Protein Kinase A-independent Ras Protein Activation Cooperates with Rap1 Protein to Mediate Activation of the Extracellular Signal-regulated Kinases (ERK) by cAMP.Adenylyl cyclase regulation in heart failure due to myocardial infarction in rats.A door opener for future research: agonist-induced β3-adrenoceptor desensitization in HEK cells but not CHO cells.Chemical suppressors of mlo-mediated powdery mildew resistance.Adenosine modulates light responses of rat retinal ganglion cell photoreceptors througha cAMP-mediated pathway.The epithelial-to-mesenchymal transition activator ZEB1 initiates a prometastatic competing endogenous RNA network.cCMP and cUMP Across the Tree of Life: From cCMP and cUMP Generators to cCMP- and cUMP-Regulated Cell Functions.Phosphorylation of Rap1 by cAMP-dependent Protein Kinase (PKA) Creates a Binding Site for KSR to Sustain ERK Activation by cAMP.Does Vidarabine Mediate Cardioprotection via Inhibition of AC5?Inhibitors of membranous adenylyl cyclases with affinity for adenosine receptors.
P2860
Q26781612-C270EB55-A46E-4CCC-80FC-B925B1A4EA81Q27023655-7DE2EE31-CF7C-41A8-9DA4-8FD5193973E3Q27311590-12F141E9-1634-42AE-B57B-ADF6BBC6A988Q28541448-F34174A6-20E0-40EF-9E42-93A07CDDC266Q30486745-DA68AC39-5C5C-46B7-994D-456F69D90245Q33806234-90F099B1-662C-45F1-9CCF-A3789A171DF3Q34640115-8B5AF323-1501-4A82-B65A-3E0C2BFAFFE9Q34760546-45C33F4B-E97F-46D0-9071-A630AF0A1472Q34906523-87BC7557-24F6-4FAD-8F7A-F9D20E1DCF59Q34978520-EED7CAEB-8E1D-4820-9B4B-5F3053F62DF7Q34979178-5F0F03F6-BEDF-4F71-BF1B-1C07325EC7C7Q35002775-62A597DD-312B-4E77-B109-9B577E29B425Q35035803-1C35E3C2-5B82-411F-8974-77E7B87FA3A4Q35543592-A0E9FCDF-C2A7-4E7B-B3D5-864FBFBB44C5Q35600378-0ADFCCCC-95AF-40D8-9C76-9C1CCC04FF18Q36144310-FA9B218A-158B-4A5D-9FAB-2479E3C4FE9BQ36287047-55473C02-D2BA-447E-9EAB-681EDAF4D32DQ36454170-4F70DAD5-6BD6-46B2-89AC-3D545BB734D4Q36497784-E533957E-20B2-4CDB-BAF3-7D67DEE97516Q36850094-21EA40DE-65D5-404F-94B1-8C59C242F2CDQ37331817-B15D2EB0-8BF2-4202-89BF-C4CB69EAEA33Q37559849-1C0DE570-F465-436F-9CF4-EEFA21A3B7DFQ38040779-1637E20B-C3A7-4DFB-8987-021CA24394BEQ38336214-9F88920D-17FC-4D5E-9CD5-4B5A068459ECQ38721985-0AD90261-0044-43F7-A44F-F11FEAC267B7Q39158851-A2C02008-0878-476D-8CAD-207920ED1227Q39354809-729E2805-4605-49E5-AC2E-09C93421323CQ40363493-E4310D7D-C1AF-4514-BFD4-43C47AD08D5AQ40503107-9F650DC1-162D-4408-AE3A-B3C7EA960368Q40997754-BBE8B9E6-265C-4673-B9D5-C59763F54F6AQ42112951-9187EB00-F80D-408E-B751-A5B9DCBC0186Q43634603-45680532-BB78-43D4-806B-12BF844F69E7Q44910331-AFB39F18-3FE6-46B7-B450-B6CAE927DB30Q47104454-7E7310F0-B148-4F33-B996-E6E69AE48907Q48093155-E52A367D-3D2D-4A48-B0E5-9521032D496AQ50087312-E2159D8E-252D-4BC9-9E09-FFD1222C3BD1Q50456694-26204C02-9528-4C90-8EAB-EB4945ED080CQ51243825-C97C0B81-7344-4967-BFBA-D7806C1D398DQ51648446-3FBD14ED-9176-4ADE-BA61-031C04FE3255Q51739948-BAA5B5CA-3EF6-4068-8C71-9455BEB71998
P2860
description
2011 nî lūn-bûn
@nan
2011年の論文
@ja
2011年論文
@yue
2011年論文
@zh-hant
2011年論文
@zh-hk
2011年論文
@zh-mo
2011年論文
@zh-tw
2011年论文
@wuu
2011年论文
@zh
2011年论文
@zh-cn
name
Inhibitors of membranous adenylyl cyclases.
@ast
Inhibitors of membranous adenylyl cyclases.
@en
type
label
Inhibitors of membranous adenylyl cyclases.
@ast
Inhibitors of membranous adenylyl cyclases.
@en
prefLabel
Inhibitors of membranous adenylyl cyclases.
@ast
Inhibitors of membranous adenylyl cyclases.
@en
P2093
P2860
P1476
Inhibitors of membranous adenylyl cyclases.
@en
P2093
Andreas Gille
Gerald H Lushington
Roland Seifert
Stephen R Sprang
Tung-Chung Mou
P2860
P356
10.1016/J.TIPS.2011.10.006
P577
2011-11-17T00:00:00Z