(N)-methanocarba-2MeSADP (MRS2365) is a subtype-specific agonist that induces rapid desensitization of the P2Y1 receptor of human platelets.
about
Attenuation of apoptosis in vitro and ischemia/reperfusion injury in vivo in mouse skeletal muscle by P2Y6 receptor activation.Activation of distinct P2Y receptor subtypes stimulates insulin secretion in MIN6 mouse pancreatic beta cells.Pharmacochemistry of the platelet purinergic receptors.P2Y nucleotide receptors: promise of therapeutic applicationsSer352 and Ser354 in the carboxyl terminus of the human P2Y(1) receptor are required for agonist-promoted phosphorylation and internalization in MDCK cellsDevelopment of selective high affinity antagonists, agonists, and radioligands for the P2Y1 receptor.Quantification of recombinant and platelet P2Y(1) receptors utilizing a [(125)I]-labeled high-affinity antagonist 2-iodo-N(6)-methyl-(N)-methanocarba-2'-deoxyadenosine-3',5'-bisphosphate ([(125)I]MRS2500)Caged agonist of P2Y1 and P2Y12 receptors for light-directed facilitation of platelet aggregation.Synthesis of ethyl (1S,2R,3S,4S,5S)-2,3-O-(isopropylidene)-4-hydroxy-bicyclo[3.1.0]hexane-carboxylate from L-ribose: a versatile chiral synthon for preparation of adenosine and P2 receptor ligands.Pharmacological characterization of purinergic inhibitory neuromuscular transmission in the human colon.
P2860
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P2860
(N)-methanocarba-2MeSADP (MRS2365) is a subtype-specific agonist that induces rapid desensitization of the P2Y1 receptor of human platelets.
description
2006 nî lūn-bûn
@nan
2006年の論文
@ja
2006年論文
@yue
2006年論文
@zh-hant
2006年論文
@zh-hk
2006年論文
@zh-mo
2006年論文
@zh-tw
2006年论文
@wuu
2006年论文
@zh
2006年论文
@zh-cn
name
(N)-methanocarba-2MeSADP (MRS2 ...... 1 receptor of human platelets.
@ast
(N)-methanocarba-2MeSADP (MRS2 ...... 1 receptor of human platelets.
@en
type
label
(N)-methanocarba-2MeSADP (MRS2 ...... 1 receptor of human platelets.
@ast
(N)-methanocarba-2MeSADP (MRS2 ...... 1 receptor of human platelets.
@en
prefLabel
(N)-methanocarba-2MeSADP (MRS2 ...... 1 receptor of human platelets.
@ast
(N)-methanocarba-2MeSADP (MRS2 ...... 1 receptor of human platelets.
@en
P2093
P2860
P1476
(N)-methanocarba-2MeSADP (MRS2 ...... 1 receptor of human platelets.
@en
P2093
D M Bourdon
K A Jacobson
S K Mahanty
T K Harden
P2860
P304
P356
10.1111/J.1538-7836.2006.01866.X
P577
2006-04-01T00:00:00Z