SAR Development of Lysine-Based Irreversible Inhibitors of Transglutaminase 2 for Huntington's Disease
about
An NMR-Guided Screening Method for Selective Fragment Docking and Synthesis of a Warhead Inhibitor.Transglutaminse 2 and EGGL, the protein cross-link formed by transglutaminse 2, as therapeutic targets for disabilities of old age.Transglutaminase inhibitors: a patent review.Strategies towards in vivo imaging of active transglutaminase type 2 using positron emission tomography.A fluorescence anisotropy-based assay for determining the activity of tissue transglutaminase.Synthesis and Kinetic Characterisation of Water-Soluble Fluorogenic Acyl Donors for Transglutaminase 2.In vivo evaluation of two tissue transglutaminase PET tracers in an orthotopic tumour xenograft model.
P2860
Q36083038-1A42ED63-829F-4B84-B7D3-B8C5A9FA0CF5Q37406648-08BB3213-7C41-49A3-AF1C-4FC514B4AADBQ38631307-98C2F352-9B12-4478-BB54-DC732C886190Q38886629-4A24EA51-0C7C-4C10-96C9-561BEA639BEBQ53174521-94EC5C1D-0E7E-4BB5-9114-694106EE3094Q53764493-BB156FC0-F3F1-4FDF-9A56-62BD19C6397CQ55030374-AC453886-A1B8-4245-A3E8-1A27D6821251
P2860
SAR Development of Lysine-Based Irreversible Inhibitors of Transglutaminase 2 for Huntington's Disease
description
2012 nî lūn-bûn
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2012年の論文
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2012年学术文章
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2012年学术文章
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2012年学术文章
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2012年学术文章
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2012年学术文章
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2012年學術文章
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2012年學術文章
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2012年學術文章
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name
SAR Development of Lysine-Base ...... ase 2 for Huntington's Disease
@en
SAR Development of Lysine-Base ...... se 2 for Huntington's Disease.
@nl
type
label
SAR Development of Lysine-Base ...... ase 2 for Huntington's Disease
@en
SAR Development of Lysine-Base ...... se 2 for Huntington's Disease.
@nl
prefLabel
SAR Development of Lysine-Base ...... ase 2 for Huntington's Disease
@en
SAR Development of Lysine-Base ...... se 2 for Huntington's Disease.
@nl
P2093
P2860
P356
P1476
SAR Development of Lysine-Base ...... ase 2 for Huntington's Disease
@en
P2093
Anna Pedret-Dunn
Celia Dominguez
Darshan Vaidya
Douglas Macdonald
Frederick A Brookfield
Ignacio Muñoz-Sanjuan
John Wityak
Laura Reed
Maria Beconi
P2860
P304
P356
10.1021/ML300241M
P577
2012-10-04T00:00:00Z