Antagonist action of progesterone at σ-receptors in the modulation of voltage-gated sodium channels
about
The σ2 receptor: a novel protein for the imaging and treatment of cancer.S2R(Pgrmc1): the cytochrome-related sigma-2 receptor that regulates lipid and drug metabolism and hormone signaling.Sigma-1 receptor agonists directly inhibit Nav1.2/1.4 channels.Ether modifications to 1-[2-(3,4-dimethoxyphenyl)ethyl]-4-(3-phenylpropyl)piperazine (SA4503): effects on binding affinity and selectivity for sigma receptors and monoamine transporters.The Sigma-1 Receptor as a Pluripotent Modulator in Living Systems.Novel substrates for, and sources of, progestogens for reproduction.The sigma-1 receptor binds to the Nav1.5 voltage-gated Na+ channel with 4-fold symmetry.Lack of sigma-1 receptor exacerbates ALS progression in miceProgesterone antagonism of neurite outgrowth depends on microglial activation via Pgrmc1/S2R.Progesterone Receptor Membrane Component 1 (PGRMC1) Expression in Murine RetinaSigma receptors [σRs]: biology in normal and diseased statesPgrmc1: new roles in the microglial mediation of progesterone-antagonism of estradiol-dependent neurite sprouting and in microglial activation.Nonclassical progesterone signalling molecules in the nervous system.The sigma-1 receptor: a regulator of cancer cell electrical plasticity?Development of sigma-1 (σ1) receptor fluorescent ligands as versatile tools to study σ1 receptors.Sigma-1 receptors modulate neonatal Nav1.5 ion channels in breast cancer cell lines.Pharmacological Modulation of the Sigma 1 Receptor and the Treatment of Pain.Evidences for antinociceptive effect of 17-α-hydroxyprogesterone caproate in carpal tunnel syndrome.Potential independent action of sigma receptor ligands through inhibition of the Kv2.1 channel.A direct interaction between the sigma-1 receptor and the hERG voltage-gated K+ channel revealed by atomic force microscopy and homogeneous time-resolved fluorescence (HTRF®).Sigma Receptor Binding Assays.Cocaine Effects on Dopaminergic Transmission Depend on a Balance between Sigma-1 and Sigma-2 Receptor Expression.Synthesis, radiolabelling, and evaluation of [11C]PB212 as a radioligand for imaging sigma-1 receptors using PET.Sigma-1 Receptor and Pain.
P2860
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P2860
Antagonist action of progesterone at σ-receptors in the modulation of voltage-gated sodium channels
description
2011 nî lūn-bûn
@nan
2011 թուականի Փետրուարին հրատարակուած գիտական յօդուած
@hyw
2011 թվականի փետրվարին հրատարակված գիտական հոդված
@hy
2011年の論文
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2011年学术文章
@wuu
2011年学术文章
@zh-cn
2011年学术文章
@zh-hans
2011年学术文章
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2011年学术文章
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2011年學術文章
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name
Antagonist action of progester ...... voltage-gated sodium channels
@ast
Antagonist action of progester ...... voltage-gated sodium channels
@en
Antagonist action of progester ...... voltage-gated sodium channels
@nl
type
label
Antagonist action of progester ...... voltage-gated sodium channels
@ast
Antagonist action of progester ...... voltage-gated sodium channels
@en
Antagonist action of progester ...... voltage-gated sodium channels
@nl
prefLabel
Antagonist action of progester ...... voltage-gated sodium channels
@ast
Antagonist action of progester ...... voltage-gated sodium channels
@en
Antagonist action of progester ...... voltage-gated sodium channels
@nl
P2093
P2860
P1476
Antagonist action of progester ...... voltage-gated sodium channels
@en
P2093
Arnold E Ruoho
Dominique Fontanilla
Meyer B Jackson
Molly Johannessen
Timur Mavlyutov
P2860
P304
P356
10.1152/AJPCELL.00383.2010
P407
P577
2011-02-01T00:00:00Z