Small-molecule inhibition of BRDT for male contraception. - Wikidata - wikimedia - TriplyDB

Small-molecule inhibition of BRDT for male contraception.

Small-molecule inhibition of BRDT for male contraception.

http://www.wikidata.org/entity/Q24616901

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Structural insights into recognition of acetylated histone ligands by the BRPF1 bromodomain Spermatid head elongation with normal nuclear shaping requires ADP-ribosyltransferase PARP11 (ARTD11) in mice Epigenetic regulation of the histone-to-protamine transition during spermiogenesis Manipulation of the host protein acetylation network by human immunodeficiency virus type 1 Sperm nuclear proteome and its epigenetic potential Male contraception Partners in crime: The role of tandem modules in gene transcription The bromodomain: from epigenome reader to druggable target Protein lysine acetylation by p300/CBP Mouse BAZ1A (ACF1) is dispensable for double-strand break repair but is essential for averting improper gene expression during spermatogenesis Human X-linked Intellectual Disability Factor CUL4B Is Required for Post-meiotic Sperm Development and Male Fertility.Cyclin-Dependent Kinase Inhibitor Dinaciclib Interacts with the Acetyl-Lysine Recognition Site of Bromodomains RVX-208, an inhibitor of BET transcriptional regulators with selectivity for the second bromodomain Acetyl-lysine Binding Site of Bromodomain-Containing Protein 4 (BRD4) Interacts with Diverse Kinase Inhibitors Structure-Based Design of γ-Carboline Analogues as Potent and Specific BET Bromodomain Inhibitors NMR Fragment Screening Hit Induces Plasticity of BRD7/9 Bromodomains The Bromodomain and Extra-Terminal Domain (BET) Family: Functional Anatomy of BET Paralogous Proteins Targeting bromodomains: epigenetic readers of lysine acetylation The mechanisms behind the therapeutic activity of BET bromodomain inhibition Differential diagnosis of azoospermia with proteomic biomarkers ECM1 and TEX101 quantified in seminal plasma An In-Depth Comparison of Latency-Reversing Agent Combinations in Various In Vitro and Ex Vivo HIV-1 Latency Models Identified Bryostatin-1+JQ1 and Ingenol-B+JQ1 to Potently Reactivate Viral Gene Expression The methyltransferase SMYD3 mediates the recruitment of transcriptional cofactors at the myostatin and c-Met genes and regulates skeletal muscle atrophy Bromodomain-dependent stage-specific male genome programming by Brdt Identification of novel potent human testis-specific and bromodomain-containing protein (BRDT) inhibitors using crystal structure-based virtual screening Sodium-hydrogen exchanger NHA1 and NHA2 control sperm motility and male fertility BET bromodomain proteins and epigenetic regulation of inflammation: implications for type 2 diabetes and breast cancer.Seeding collaborations to advance kinase science with the GSK Published Kinase Inhibitor Set (PKIS)Male contraception via simultaneous knockout of α1A-adrenoceptors and P2X1-purinoceptors in mice.NSD3-NUT fusion oncoprotein in NUT midline carcinoma: implications for a novel oncogenic mechanism.Characterization of BRD4 during mammalian postmeiotic sperm development.The polar warhead of a TRIM24 bromodomain inhibitor rearranges a water-mediated interaction network.Privileged diazepine compounds and their emergence as bromodomain inhibitors.The BET protein FSH functionally interacts with ASH1 to orchestrate global gene activity in Drosophila.The bromodomain inhibitor JQ1 triggers growth arrest and apoptosis in testicular germ cell tumours in vitro and in vivo.BET Inhibitor JQ1 Blocks Inflammation and Bone Destruction.Bromodomain 4 protein is a predictor of survival for urothelial carcinoma of bladder.Inhibition of BET bromodomain targets genetically diverse glioblastoma BET bromodomains mediate transcriptional pause release in heart failure Protein acetylation and spermatogenesis.BET bromodomain inhibitors: a patent review.

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Small-molecule inhibition of BRDT for male contraception.

http://www.wikidata.org/entity/Q24616901

description

2012 nî lūn-bûn

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2012 թուականի Օգոստոսին հրատարակուած գիտական յօդուած

@hyw

2012 թվականի օգոստոսին հրատարակված գիտական հոդված

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2012年の論文

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2012年学术文章

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2012年学术文章

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2012年学术文章

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2012年学术文章

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2012年学术文章

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2012年學術文章

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name

Small-molecule inhibition of BRDT for male contraception

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Small-molecule inhibition of BRDT for male contraception.

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Small-molecule inhibition of BRDT for male contraception.

@en

type

label

Small-molecule inhibition of BRDT for male contraception

@nl

Small-molecule inhibition of BRDT for male contraception.

@ast

Small-molecule inhibition of BRDT for male contraception.

@en

altLabel

Small-Molecule Inhibition of BRDT for Male Contraception

@en

prefLabel

Small-molecule inhibition of BRDT for male contraception

@nl

Small-molecule inhibition of BRDT for male contraception.

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Small-molecule inhibition of BRDT for male contraception.

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Small-molecule inhibition of BRDT for male contraception.

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Julio E Agno

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Jun Qi

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Lang Ma

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Martin M Matzuk

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Richard N Yu

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Sarah Picaud

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P2860

Cyclin A1 is required for meiosis in the male mouse

Structure and ligand of a histone acetyltransferase bromodomain

Selective inhibition of BET bromodomains

Gene set enrichment analysis: a knowledge-based approach for interpreting genome-wide expression profiles.

MAFFT: a novel method for rapid multiple sequence alignment based on fast Fourier transform

MAFFT version 5: improvement in accuracy of multiple sequence alignment

As the world grows: contraception in the 21st century

An integrated database of genes responsive to the Myc oncogenic transcription factor: identification of direct genomic targets

Cooperative binding of two acetylation marks on a histone tail by a single bromodomain

Suppression of inflammation by a synthetic histone mimic

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Panagis Filippakopoulos

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