Characterization of [(125)I]-SB-258585 binding to human recombinant and native 5-HT(6) receptors in rat, pig and human brain tissue
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SB-656104-A, a novel selective 5-HT7 receptor antagonist, modulates REM sleep in ratsExpression of serotonin 5-HT(2A) receptors in the human cerebellum and alterations in schizophrenia.5-HT6 receptor binding sites in schizophrenia and following antipsychotic drug administration: autoradiographic studies with [125I]SB-258585.5-HT radioligands for human brain imaging with PET and SPECTThe 5-HT(6) receptor antagonist SB-271046 reverses scopolamine-disrupted consolidation of a passive avoidance task and ameliorates spatial task deficits in aged rats.Binding of serotonin and N1-benzenesulfonyltryptamine-related analogs at human 5-HT6 serotonin receptors: receptor modeling studies.Characterization of SB-271046: a potent, selective and orally active 5-HT(6) receptor antagonistPET tracers for serotonin receptors and their applicationsDeconstructing 5-HT6 receptor effects on striatal circuit function.Measuring endogenous 5-HT release by emission tomography: promises and pitfalls.The serotonin-6 receptor as a novel therapeutic target.Considerations in the Development of Reversibly Binding PET Radioligands for Brain Imaging.Characterization and Reliability of [18F]2FNQ1P in Cynomolgus Monkeys as a PET Radiotracer for Serotonin 5-HT6 Receptors.Differential involvement of 5-HT(1B/1D) and 5-HT6 receptors in cognitive and non-cognitive symptoms in Alzheimer's disease.Excess of serotonin affects embryonic interneuron migration through activation of the serotonin receptor 6.A comparison of multiple 5-HT receptors in two tasks measuring impulsivity.Design, synthesis and pharmacological evaluation of indolylsulfonamide amines as potent and selective 5-HT6 receptor antagonists.MDMA induces EPSP-Spike potentiation in rat ventral hippocampus in vitro via serotonin and noradrenaline release and coactivation of 5-HT4 and beta1 receptors.Preclinical evaluation of [18F]2FNQ1P as the first fluorinated serotonin 5-HT6 radioligand for PET imaging.Distribution of serotonin receptor of type 6 (5-HT₆) in human brain post-mortem. A pharmacology, autoradiography and immunohistochemistry study.Synthesis and biological evaluation of novel N1-phenylsulphonyl indole derivatives as potent and selective 5-HT6R ligands for the treatment of cognitive disorders.Extended N-Arylsulfonylindoles as 5-HT₆ Receptor Antagonists: Design, Synthesis & Biological Evaluation.
P2860
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P2860
Characterization of [(125)I]-SB-258585 binding to human recombinant and native 5-HT(6) receptors in rat, pig and human brain tissue
description
2000 nî lūn-bûn
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2000 թուականի Օգոստոսին հրատարակուած գիտական յօդուած
@hyw
2000 թվականի օգոստոսին հրատարակված գիտական հոդված
@hy
2000年の論文
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2000年論文
@yue
2000年論文
@zh-hant
2000年論文
@zh-hk
2000年論文
@zh-mo
2000年論文
@zh-tw
2000年论文
@wuu
name
Characterization of [(125)I]-S ...... at, pig and human brain tissue
@ast
Characterization of [(125)I]-S ...... at, pig and human brain tissue
@en
Characterization of [(125)I]-S ...... at, pig and human brain tissue
@nl
type
label
Characterization of [(125)I]-S ...... at, pig and human brain tissue
@ast
Characterization of [(125)I]-S ...... at, pig and human brain tissue
@en
Characterization of [(125)I]-S ...... at, pig and human brain tissue
@nl
prefLabel
Characterization of [(125)I]-S ...... at, pig and human brain tissue
@ast
Characterization of [(125)I]-S ...... at, pig and human brain tissue
@en
Characterization of [(125)I]-S ...... at, pig and human brain tissue
@nl
P2093
P2860
P356
P1476
Characterization of [(125)I]-S ...... at, pig and human brain tissue
@en
P2093
A J Latter
C Routledge
D N Middlemiss
J A Minton
S M Bromidge
P2860
P304
P356
10.1038/SJ.BJP.0703458
P407
P577
2000-08-01T00:00:00Z