Discoidin domain receptor 1 (DDR1) kinase as target for structure-based drug discovery
about
Discoidin Domain Receptors: Potential Actors and Targets in CancerHMGB1 induces apoptosis and EMT in association with increased autophagy following H/R injury in cardiomyocytesIGF-I induces upregulation of DDR1 collagen receptor in breast cancer cells by suppressing MIR-199a-5p through the PI3K/AKT pathway.Structure-Based Design of Tetrahydroisoquinoline-7-carboxamides as Selective Discoidin Domain Receptor 1 (DDR1) Inhibitors.Analogs, formulations and derivatives of imatinib: a patent review.Synthesis and biological evaluation of novel dasatinib analogues as potent DDR1 and DDR2 kinase inhibitors.Contribution of collagen adhesion receptors to tissue fibrosis.Harnessing the power of proteomics for identification of oncogenic, druggable signalling pathways in cancer.Discoidin domain receptor 1 kinase activity is required for regulating collagen IV synthesis.Identification of novel inhibitors of DDR1 against idiopathic pulmonary fibrosis by integrative transcriptome meta-analysis, computational and experimental screening.
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Q26751157-B68A1024-7A1B-4D0F-AED2-3ABF5EC6A7B7Q36630684-E284361A-F964-4342-B11C-1567257FCCCDQ36946586-D7738EB1-9F9A-47FC-BA14-651296812734Q37317054-BD54B8C4-8640-43C4-8CB7-C654111F7F5BQ38587332-5F5CCE2B-7B8D-4BEF-8E5F-05A5CFDA2A74Q38748552-45D60CB6-29CF-4C0A-9A2F-67BFF6B6B294Q38879377-F3A4FEE0-A40A-44FA-955A-8D4AA1075F38Q39175714-5F6F190D-4050-4343-BF10-88F47D7F88CDQ48021722-25D149E9-763C-4C6D-A218-E93AE8D37A65Q55026945-8157A0A6-72B4-44BA-B18C-1BCC8C36AB50
P2860
Discoidin domain receptor 1 (DDR1) kinase as target for structure-based drug discovery
description
2015 nî lūn-bûn
@nan
2015 թուականի Փետրուարին հրատարակուած գիտական յօդուած
@hyw
2015 թվականի փետրվարին հրատարակված գիտական հոդված
@hy
2015年の論文
@ja
2015年論文
@yue
2015年論文
@zh-hant
2015年論文
@zh-hk
2015年論文
@zh-mo
2015年論文
@zh-tw
2015年论文
@wuu
name
Discoidin domain receptor 1 (DDR1) kinase as target for structure-based drug discovery
@ast
Discoidin domain receptor 1 (DDR1) kinase as target for structure-based drug discovery
@en
Discoidin domain receptor 1 (DDR1) kinase as target for structure-based drug discovery
@nl
type
label
Discoidin domain receptor 1 (DDR1) kinase as target for structure-based drug discovery
@ast
Discoidin domain receptor 1 (DDR1) kinase as target for structure-based drug discovery
@en
Discoidin domain receptor 1 (DDR1) kinase as target for structure-based drug discovery
@nl
prefLabel
Discoidin domain receptor 1 (DDR1) kinase as target for structure-based drug discovery
@ast
Discoidin domain receptor 1 (DDR1) kinase as target for structure-based drug discovery
@en
Discoidin domain receptor 1 (DDR1) kinase as target for structure-based drug discovery
@nl
P2093
P2860
P3181
P1433
P1476
Discoidin domain receptor 1 (DDR1) kinase as target for structure-based drug discovery
@en
P2093
Ambra Pozzi
Corina M. Borza
Edward W. Lowe
Sandeepkumar Kothiwale
P2860
P304
P3181
P356
10.1016/J.DRUDIS.2014.09.025
P407
P50
P577
2015-02-01T00:00:00Z