Anilinoquinazoline inhibitors of fructose 1,6-bisphosphatase bind at a novel allosteric site: synthesis, in vitro characterization, and X-ray crystallography

Anilinoquinazoline inhibitors of fructose 1,6-bisphosphatase bind at a novel allosteric site: synthesis, in vitro characterization, and X-ray crystallography

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http://www.wikidata.org/entity/Q27639512
Metaphosphate in the active site of fructose-1,6-bisphosphataseInhibition of fructose-1,6-bisphosphatase by a new class of allosteric effectorsStructures of mammalian and bacterial fructose-1,6-bisphosphatase reveal the basis for synergism in AMP/fructose 2,6-bisphosphate inhibitionStructural and Biochemical Characterization of the Type II Fructose-1,6-bisphosphatase GlpX from Escherichia coliCrystal structures of Plasmodium falciparum cytosolic tryptophanyl-tRNA synthetase and its potential as a target for structure-guided drug designA library of novel allosteric inhibitors against fructose 1,6-bisphosphatase.Structure-based predictive models for allosteric hot spots.MB06322 (CS-917): A potent and selective inhibitor of fructose 1,6-bisphosphatase for controlling gluconeogenesis in type 2 diabetes.Designing inhibitors against fructose 1,6-bisphosphatase: exploring natural products for novel inhibitor scaffoldsIn silico identification of structure requirement for novel thiazole and oxazole derivatives as potent fructose 1,6-bisphosphatase inhibitors.Recent advances in the design and synthesis of prazosin derivatives.Quadruple space-group ambiguity owing to rotational and translational noncrystallographic symmetry in human liver fructose-1,6-bisphosphatase.Toward the prediction of FBPase inhibitory activity using chemoinformatic methods.An integrative in-silico approach for therapeutic target identification in the human pathogen Corynebacterium diphtheriae.Elucidation of direct competition and allosteric modulation of small-molecular-weight protein ligands using surface plasmon resonance methods.The Druggable Pocketome of Corynebacterium diphtheriae: A New Approach for in silico Putative Druggable Targets.Reversing allosteric communication: From detecting allosteric sites to inducing and tuning targeted allosteric response.
P2860

Anilinoquinazoline inhibitors of fructose 1,6-bisphosphatase bind at a novel allosteric site: synthesis, in vitro characterization, and X-ray crystallography

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http://www.wikidata.org/entity/Q27639512
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2002 nî lūn-bûn
@nan
2002 թուականի Օգոստոսին հրատարակուած գիտական յօդուած
@hyw
2002 թվականի օգոստոսին հրատարակված գիտական հոդված
@hy
2002年の論文
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2002年学术文章
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2002年学术文章
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2002年学术文章
@zh-hans
2002年学术文章
@zh-my
2002年学术文章
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2002年學術文章
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name
Anilinoquinazoline inhibitors ...... ion, and X-ray crystallography
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Anilinoquinazoline inhibitors ...... ion, and X-ray crystallography
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Anilinoquinazoline inhibitors ...... ion, and X-ray crystallography
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type
label
Anilinoquinazoline inhibitors ...... ion, and X-ray crystallography
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Anilinoquinazoline inhibitors ...... ion, and X-ray crystallography
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Anilinoquinazoline inhibitors ...... ion, and X-ray crystallography
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prefLabel
Anilinoquinazoline inhibitors ...... ion, and X-ray crystallography
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Anilinoquinazoline inhibitors ...... ion, and X-ray crystallography
@en
Anilinoquinazoline inhibitors ...... ion, and X-ray crystallography
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P1433
P1476
P2093
P304
P31
P356
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P433
P478
P50
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P921
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P1433
P1476
Anilinoquinazoline inhibitors ...... ion, and X-ray crystallography
@en
P2093
P304
P31
P356
P407
P433
P478
P50
P577
P698
P921