X-ray Structures of Human Furin in Complex with Competitive Inhibitors
about
K153R polymorphism in myostatin gene increases the rate of promyostatin activation by furinNovel Furin Inhibitors with Potent Anti-infectious ActivityEbola virus: A gap in drug design and discovery - experimental and computational perspective.Identification of potent and compartment-selective small molecule furin inhibitors using cell-based assays.Structure and stabilization of the Hendra virus F glycoprotein in its prefusion formThe structure of a furin-antibody complex explains non-competitive inhibition by steric exclusion of substrate conformers.Structure of the unliganded form of the proprotein convertase furin suggests activation by a substrate-induced mechanism.Therapeutic uses of furin and its inhibitors: a patent review.PACE4 inhibitors and their peptidomimetic analogs block prostate cancer tumor progression through quiescence induction, increased apoptosis and impaired neovascularisation.Human furin Cys198 imposes dihedral and positional restraints on His194 for optimal Ser386-proton transfer.The proprotein convertase furin in tumour progression.Ebola virus envelope glycoprotein derived peptide in human Furin-bound state: computational studies.Elongated and Shortened Peptidomimetic Inhibitors of the Proprotein Convertase Furin.Chemical structure and properties of low-molecular furin inhibitors.Optimization of Substrate-Analogue Furin Inhibitors.Rational Design of a Highly Potent and Selective Peptide Inhibitor of PACE4 by Salt Bridge Interaction with D160 at Position P3.Engineering a Constrained Peptidic Scaffold towards Potent and Selective Furin Inhibitors.
P2860
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P2860
X-ray Structures of Human Furin in Complex with Competitive Inhibitors
description
2014 nî lūn-bûn
@nan
2014 թուականի Մայիսին հրատարակուած գիտական յօդուած
@hyw
2014 թվականի մայիսին հրատարակված գիտական հոդված
@hy
2014年の論文
@ja
2014年論文
@yue
2014年論文
@zh-hant
2014年論文
@zh-hk
2014年論文
@zh-mo
2014年論文
@zh-tw
2014年论文
@wuu
name
X-ray Structures of Human Furin in Complex with Competitive Inhibitors
@ast
X-ray Structures of Human Furin in Complex with Competitive Inhibitors
@en
X-ray Structures of Human Furin in Complex with Competitive Inhibitors
@nl
type
label
X-ray Structures of Human Furin in Complex with Competitive Inhibitors
@ast
X-ray Structures of Human Furin in Complex with Competitive Inhibitors
@en
X-ray Structures of Human Furin in Complex with Competitive Inhibitors
@nl
prefLabel
X-ray Structures of Human Furin in Complex with Competitive Inhibitors
@ast
X-ray Structures of Human Furin in Complex with Competitive Inhibitors
@en
X-ray Structures of Human Furin in Complex with Competitive Inhibitors
@nl
P2093
P2860
P3181
P356
P1433
P1476
X-ray structures of human furin in complex with competitive inhibitors
@en
P2093
Gero L Becker
Kornelia Hardes
Manuel E Than
Torsten Steinmetzer
P2860
P304
P3181
P356
10.1021/CB500087X
P577
2014-04-01T00:00:00Z