Pharmacological and biochemical analysis of FPL 67156, a novel, selective inhibitor of ecto-ATPase
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Local regulation of [(3)H]-noradrenaline release from the isolated guinea-pig right atrium by P(2X)-receptors located on axon terminalsLeishmania infantum ecto-nucleoside triphosphate diphosphohydrolase-2 is an apyrase involved in macrophage infection and expressed in infected dogsThe expression level of ecto-NTP diphosphohydrolase1/CD39 modulates exocytotic and ischemic release of neurotransmitters in a cellular model of sympathetic neuronsPlasmodium falciparum GFP-E-NTPDase expression at the intraerythrocytic stages and its inhibition blocks the development of the human malaria parasiteInfluence of Ecto-nucleoside triphosphate diphosphohydrolase activity on Trypanosoma cruzi infectivity and virulenceATP-gated P2X3 receptors constitute a positive autocrine signal for insulin release in the human pancreatic beta cellTiclopidine in its prodrug form is a selective inhibitor of human NTPDase1Increased CD39 nucleotidase activity on microparticles from patients with idiopathic pulmonary arterial hypertension.E-NTPDase1/CD39 modulates renin release from heart mast cells during ischemia/reperfusion: a novel cardioprotective role.The GDA1_CD39 superfamily: NTPDases with diverse functions.ATP, a partial agonist for the P2Z receptor of human lymphocytesCharacterization of the ATPase released during sympathetic nerve stimulation of the guinea-pig isolated vas deferensRelease of a soluble ATPase from the rabbit isolated vas deferens during nerve stimulationMethylene ATP analogs as modulators of extracellular ATP metabolism and accumulation.Evidence for two distinct P2-purinoceptors subserving contraction of the rat anococcygeus smooth muscleInhibition of ecto-ATPase by PPADS, suramin and reactive blue in endothelial cells, C6 glioma cells and RAW 264.7 macrophagesPyrimidinoceptor-mediated activation of phospholipase C and phospholipase A2 in RAW 264.7 macrophages.Metabolism of circulating ADP in the bloodstream is mediated via integrated actions of soluble adenylate kinase-1 and NTPDase1/CD39 activitiesRelative contribution of ecto-ATPase and ecto-ATPDase pathways to the biphasic effect of ATP on acetylcholine release from myenteric motoneurons.Purinergic signalling in the urinary tract in health and disease.Therapeutic potentials of ecto-nucleoside triphosphate diphosphohydrolase, ecto-nucleotide pyrophosphatase/phosphodiesterase, ecto-5'-nucleotidase, and alkaline phosphatase inhibitors.Generation and characterization of polyclonal and monoclonal antibodies to human NTPDase2 including a blocking antibody.P2-purinoceptor-mediated formation of inositol phosphates and intracellular Ca2+ transients in human coronary artery smooth muscle cellsEctonucleotidases CD39 and CD73 on OvCA cells are potent adenosine-generating enzymes responsible for adenosine receptor 2A-dependent suppression of T cell function and NK cell cytotoxicity.Astrocyte cultures exhibit P2X7 receptor channel opening in the absence of exogenous ligands.Ectonucleotidases in Müller glial cells of the rodent retina: Involvement in inhibition of osmotic cell swelling.Selective nucleoside triphosphate diphosphohydrolase-2 (NTPDase2) inhibitors: nucleotide mimetics derived from uridine-5'-carboxamide.8-BuS-ATP derivatives as specific NTPDase1 inhibitors.Auto-inhibition of rat parallel fibre-Purkinje cell synapses by activity-dependent adenosine release.Control of basal extracellular adenosine concentration in rat cerebellum.Degradation of extracellular ATP by the retinal pigment epithelium.A capillary electrophoresis method for the characterization of ecto-nucleoside triphosphate diphosphohydrolases (NTPDases) and the analysis of inhibitors by in-capillary enzymatic microreaction.Role of P2 purinergic receptors in synaptic transmission under normoxic and ischaemic conditions in the CA1 region of rat hippocampal slices.Kinetics of ATP release following compression injury of a peripheral nerve trunk.A commonly used ecto-ATPase inhibitor, ARL-67156, blocks degradation of ADP more than the degradation of ATP in murine colonPPADS and suramin as antagonists at cloned P2Y- and P2U-purinoceptors.Purinoceptors: from history to recent progress. A review.Extracellular metabolism of nucleotides in the nervous system.Ecto-nucleoside triphosphate diphosphohydrolase 1 (E-NTPDase1/CD39) regulates neutrophil chemotaxis by hydrolyzing released ATP to adenosine.High affinity P2x-purinoceptor binding sites for [35S]-adenosine 5'-O-[3-thiotriphosphate] in rat vas deferens membranes.
P2860
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P2860
Pharmacological and biochemical analysis of FPL 67156, a novel, selective inhibitor of ecto-ATPase
description
1995 nî lūn-bûn
@nan
1995 թուականի Յունուարին հրատարակուած գիտական յօդուած
@hyw
1995 թվականի հունվարին հրատարակված գիտական հոդված
@hy
1995年の論文
@ja
1995年論文
@yue
1995年論文
@zh-hant
1995年論文
@zh-hk
1995年論文
@zh-mo
1995年論文
@zh-tw
1995年论文
@wuu
name
Pharmacological and biochemica ...... ctive inhibitor of ecto-ATPase
@ast
Pharmacological and biochemica ...... ctive inhibitor of ecto-ATPase
@en
Pharmacological and biochemica ...... ctive inhibitor of ecto-ATPase
@nl
type
label
Pharmacological and biochemica ...... ctive inhibitor of ecto-ATPase
@ast
Pharmacological and biochemica ...... ctive inhibitor of ecto-ATPase
@en
Pharmacological and biochemica ...... ctive inhibitor of ecto-ATPase
@nl
prefLabel
Pharmacological and biochemica ...... ctive inhibitor of ecto-ATPase
@ast
Pharmacological and biochemica ...... ctive inhibitor of ecto-ATPase
@en
Pharmacological and biochemica ...... ctive inhibitor of ecto-ATPase
@nl
P2093
P2860
P1476
Pharmacological and biochemica ...... ctive inhibitor of ecto-ATPase
@en
P2093
A H Ingall
A P IJzerman
C E Pollard
K C McKechnie
M W Beukers
S M Roberts
P2860
P304
P356
10.1111/J.1476-5381.1995.TB13251.X
P407
P577
1995-01-01T00:00:00Z