Inhibition of human immunodeficiency virus integrase by bis-catechols
about
A historical sketch of the discovery and development of HIV-1 integrase inhibitorsResistance to the anti-human immunodeficiency virus type 1 compound L-chicoric acid results from a single mutation at amino acid 140 of integraseHuman immunodeficiency virus type 1 cDNA integration: new aromatic hydroxylated inhibitors and studies of the inhibition mechanism.Isolation and characterization of novel human immunodeficiency virus integrase inhibitors from fungal metabolitesIdentification of a hexapeptide inhibitor of the human immunodeficiency virus integrase protein by using a combinatorial chemical libraryInhibitors of HIV-1 replication [corrected; erratum to be published] that inhibit HIV integraseDifferential inhibition of HIV-1 preintegration complexes and purified integrase protein by small moleculesDicaffeoylquinic and dicaffeoyltartaric acids are selective inhibitors of human immunodeficiency virus type 1 integrase.Equivalent inhibition of half-site and full-site retroviral strand transfer reactions by structurally diverse compoundsInhibition of acute-, latent-, and chronic-phase human immunodeficiency virus type 1 (HIV-1) replication by a bistriazoloacridone analog that selectively inhibits HIV-1 transcriptionDiarylsulfones, a novel class of human immunodeficiency virus type 1 integrase inhibitorsNucleophile selection for the endonuclease activities of human, ovine, and avian retroviral integrases.Irreversible inhibition of human immunodeficiency virus type 1 integrase by dicaffeoylquinic acids.Efficiency and fidelity of full-site integration reactions using recombinant simian immunodeficiency virus integraseCurrent developments in HIV chemotherapy.HIV integrase inhibitors as therapeutic agents in AIDS.HIV-1 integrase inhibitors: a review of their chemical development.Alternate strand DNA triple helix-mediated inhibition of HIV-1 U5 long terminal repeat integration in vitro.Effects of mutations in residues near the active site of human immunodeficiency virus type 1 integrase on specific enzyme-substrate interactions.Differential divalent cation requirements uncouple the assembly and catalytic reactions of human immunodeficiency virus type 1 integrase.Design and synthesis of novel dihydroxyindole-2-carboxylic acids as HIV-1 integrase inhibitors.Synthesis and anti-human immunodeficiency virus type 1 integrase activity of hydroxybenzoic and hydroxycinnamic acid flavon-3-yl esters.Structure-Guided Optimization of HIV Integrase Strand Transfer Inhibitors.Tricyclic flavonoids with 1,3-dithiolium substructure.
P2860
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P2860
Inhibition of human immunodeficiency virus integrase by bis-catechols
description
1995 nî lūn-bûn
@nan
1995 թուականի Փետրուարին հրատարակուած գիտական յօդուած
@hyw
1995 թվականի փետրվարին հրատարակված գիտական հոդված
@hy
1995年の論文
@ja
1995年論文
@yue
1995年論文
@zh-hant
1995年論文
@zh-hk
1995年論文
@zh-mo
1995年論文
@zh-tw
1995年论文
@wuu
name
Inhibition of human immunodeficiency virus integrase by bis-catechols
@ast
Inhibition of human immunodeficiency virus integrase by bis-catechols
@en
Inhibition of human immunodeficiency virus integrase by bis-catechols
@nl
type
label
Inhibition of human immunodeficiency virus integrase by bis-catechols
@ast
Inhibition of human immunodeficiency virus integrase by bis-catechols
@en
Inhibition of human immunodeficiency virus integrase by bis-catechols
@nl
prefLabel
Inhibition of human immunodeficiency virus integrase by bis-catechols
@ast
Inhibition of human immunodeficiency virus integrase by bis-catechols
@en
Inhibition of human immunodeficiency virus integrase by bis-catechols
@nl
P2093
P2860
P356
P1476
Inhibition of human immunodeficiency virus integrase by bis-catechols
@en
P2093
D J Hazuda
J C Hastings
P L Graham
R L LaFemina
P2860
P356
10.1128/AAC.39.2.320
P407
P577
1995-02-01T00:00:00Z