Discovery of Carbohydrate Sulfotransferase Inhibitors from a Kinase-Directed Library We thank Sharon Long and Dave Keating for providing both the NodH sulfotransferase and APS Kinase during our preliminary experiments and Jack Kirsch for numerous he
about
The Regulation of Steroid Action by Sulfation and DesulfationA structural and biochemical basis for PAPS-independent sulfuryl transfer by aryl sulfotransferase from uropathogenic Escherichia coliProtein structure similarity as guiding principle for combinatorial library design.Mass spectrometry and immobilized enzymes for the screening of inhibitor libraries.Rapid discovery of potent sulfotransferase inhibitors by diversity-oriented reaction in microplates followed by in situ screening.Inhibitory peptides of the sulfotransferase domain of the heparan sulfate enzyme, N-deacetylase-N-sulfotransferase-1.Modifications of glycans: biological significance and therapeutic opportunitiesRecent development in the design of sialyltransferase inhibitors.Drug targets in mycobacterial sulfur metabolism.New targets and inhibitors of mycobacterial sulfur metabolism.Strategies for facilitated forward chemical genetics.Recent advances in sulfotransferase enzyme activity assays.Glycan antagonists and inhibitors: a fount for drug discovery.A small-molecule switch for Golgi sulfotransferases.Drug-Mediated Regulation of Glycosaminoglycan Biosynthesis.Small-molecule inhibition of pyruvate phosphate dikinase targeting the nucleotide binding site.Trisubstituted purines are useful tools for developing potent plant mitogen-activated protein kinase inhibitors.Diversity-Based Organic Synthesis in the Era of Genomics and Proteomics NRC publication no. 43843. David Thomas is a senior colleague and mentor.New tools for carbohydrate sulfation analysis: heparan sulfate 2--sulfotransferase (HS2ST) is a target for small-molecule protein kinase inhibitorsNew tools for evaluating protein tyrosine sulfation: tyrosylprotein sulfotransferases (TPSTs) are novel targets for RAF protein kinase inhibitors
P2860
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P2860
Discovery of Carbohydrate Sulfotransferase Inhibitors from a Kinase-Directed Library We thank Sharon Long and Dave Keating for providing both the NodH sulfotransferase and APS Kinase during our preliminary experiments and Jack Kirsch for numerous he
description
2000 nî lūn-bûn
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2000 թուականի Ապրիլին հրատարակուած գիտական յօդուած
@hyw
2000 թվականի ապրիլին հրատարակված գիտական հոդված
@hy
2000年の論文
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2000年論文
@yue
2000年論文
@zh-hant
2000年論文
@zh-hk
2000年論文
@zh-mo
2000年論文
@zh-tw
2000年论文
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name
Discovery of Carbohydrate Sulf ...... nd Jack Kirsch for numerous he
@ast
Discovery of Carbohydrate Sulf ...... nd Jack Kirsch for numerous he
@en
type
label
Discovery of Carbohydrate Sulf ...... nd Jack Kirsch for numerous he
@ast
Discovery of Carbohydrate Sulf ...... nd Jack Kirsch for numerous he
@en
prefLabel
Discovery of Carbohydrate Sulf ...... nd Jack Kirsch for numerous he
@ast
Discovery of Carbohydrate Sulf ...... nd Jack Kirsch for numerous he
@en
P2093
P1476
Discovery of Carbohydrate Sulf ...... ciety (Grant No. RPG9700501BE)
@en
P2093
Armstrong JI
Bertozzi CR
Nierengarten DM
Portley AR
Schultz PG
P304
P356
10.1002/(SICI)1521-3773(20000403)39:7<1303::AID-ANIE1303>3.0.CO;2-0
P407
P577
2000-04-01T00:00:00Z