Structure-guided discovery of novel aminoglycoside mimetics as antibacterial translation inhibitors
about
Small molecule microarrays of RNA-focused peptoids help identify inhibitors of a pathogenic group I intronSearch for novel aminoglycosides by combining fragment-based virtual screening and 3D-QSAR scoring1,3-Diazepanes of natural product-like complexity from cyanamide-induced rearrangement of epoxy-delta-lactams.Hepatitis C virus translation inhibitors targeting the internal ribosomal entry site.Myxobacterium-produced antibiotic TA (myxovirescin) inhibits type II signal peptidaseSynthesis and SAR of 3,5-diamino-piperidine derivatives: novel antibacterial translation inhibitors as aminoglycoside mimetics.A modular approach to synthetic RNA binders of the hepatitis C virus internal ribosome entry site.Antibacterial activity in serum of the 3,5-diamino-piperidine translation inhibitors.Fluorescent HIV-1 Dimerization Initiation Site: design, properties, and use for ligand discoveryThemes and variations in riboswitch structure and function.Hygromycin B inhibition of protein synthesis and ribosome biogenesis in Escherichia coli.Design, synthesis, antibacterial activity, and molecular docking studies of novel hybrid 1,3-thiazine-1,3,5-triazine derivatives as potential bacterial translation inhibitor.Potential new antibiotic sites in the ribosome revealed by deleterious mutations in RNA of the large ribosomal subunit.
P2860
Q33417035-6B4A7E57-F73C-4A60-945C-E0F5A65D6B98Q33444102-63591A58-D3CE-4758-9A45-80ECB6D1B7F3Q33520303-7BE64322-A51A-4951-91EB-5CCB79B1C669Q34038589-D599045A-2608-4F6F-BDED-FF59B610BE13Q34122542-05B7BF00-48AE-4780-8CE0-3EFF7D35FCD2Q35765813-D121C27D-EDC7-4287-862F-EBC48A50A6C7Q36452979-CE328BEB-E69B-46F7-8B90-12C67FD0513CQ36775946-DC7BD366-21C4-4335-8463-70FA9D4DB2F9Q36852633-AABB97D3-1D93-43BF-A359-8B6E336EFCAFQ38192408-453F5C3E-B850-4CA8-ABBC-A6E90DE07192Q42727860-DDD248DB-A55C-4534-A93E-DAC3C7B9699AQ44589141-4031F6CB-E7F8-40F4-A34C-11D7E861EE73Q54439108-43D80943-BE18-433D-AADE-695ED0669AF5
P2860
Structure-guided discovery of novel aminoglycoside mimetics as antibacterial translation inhibitors
description
2005 nî lūn-bûn
@nan
2005 թուականի Դեկտեմբերին հրատարակուած գիտական յօդուած
@hyw
2005 թվականի դեկտեմբերին հրատարակված գիտական հոդված
@hy
2005年の論文
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2005年学术文章
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2005年学术文章
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2005年学术文章
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2005年学术文章
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2005年学术文章
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2005年學術文章
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name
Structure-guided discovery of ...... cterial translation inhibitors
@ast
Structure-guided discovery of ...... cterial translation inhibitors
@en
Structure-guided discovery of ...... cterial translation inhibitors
@nl
type
label
Structure-guided discovery of ...... cterial translation inhibitors
@ast
Structure-guided discovery of ...... cterial translation inhibitors
@en
Structure-guided discovery of ...... cterial translation inhibitors
@nl
prefLabel
Structure-guided discovery of ...... cterial translation inhibitors
@ast
Structure-guided discovery of ...... cterial translation inhibitors
@en
Structure-guided discovery of ...... cterial translation inhibitors
@nl
P2093
P2860
P1476
Structure-guided discovery of ...... cterial translation inhibitors
@en
P2093
Benjamin K Ayida
Daniel Wall
Dionisios Vourloumis
Douglas Murphy
Geoffrey C Winters
Jamie M Froelich
Klaus B Simonsen
Sarah Fish
Thomas Hermann
Vlad E Gregor
P2860
P304
P356
10.1128/AAC.49.12.4942-4949.2005
P407
P577
2005-12-01T00:00:00Z