Rhodanine as a scaffold in drug discovery: a critical review of its biological activities and mechanisms of target modulation.
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Histone-modifying enzymes, histone modifications and histone chaperones in nucleosome assembly: Lessons learned from Rtt109 histone acetyltransferasesRhodanine hydrolysis leads to potent thioenolate mediated metallo-β-lactamase inhibitionCovalent Modifiers: A Chemical Perspective on the Reactivity of α,β-Unsaturated Carbonyls with Thiols via Hetero-Michael Addition ReactionsDiscovery of Mycobacterium tuberculosis InhA Inhibitors by Binding Sites Comparison and Ligands Prediction.Crystal structure of N-(4-oxo-2-sulfanyl-idene-1,3-thia-zolidin-3-yl)-2-(thio-phen-3-yl)acetamide.The essential roles of chemistry in high-throughput screening triageSmall-molecule procaspase activators identified using fluorescence polarization.A small molecule screen identifies selective inhibitors of urea transporter UT-A.Synthesis and Anticancer Activity of New Thiopyrano[2,3-d]thiazoles Based on Cinnamic Acid Amides.Non-stoichiometric inhibition in integrated lead finding - a literature review.Inhibition of Cancer-Associated Mutant Isocitrate Dehydrogenases by 2-Thiohydantoin CompoundsQuality Issues with Public Domain Chemogenomics Data.Probing the Azaaurone Scaffold against the Hepatic and Erythrocytic Stages of Malaria Parasites.Pharmacological Chaperoning: A Potential Treatment for PMM2-CDG.The Small Molecule IMR-1 Inhibits the Notch Transcriptional Activation Complex to Suppress Tumorigenesis.Exploration of a series of 5-arylidene-2-thioxoimidazolidin-4-ones as inhibitors of the cytolytic protein perforinMultitarget ligands in antibacterial research: progress and opportunities.Viable screening targets related to the bacterial cell wall.Computational Search for Possible Mechanisms of 4-Thiazolidinones Anticancer Activity: The Power of Visualization.Furan-based benzene mono- and dicarboxylic acid derivatives as multiple inhibitors of the bacterial Mur ligases (MurC-MurF): experimental and computational characterization.Antibacterial properties of 5-substituted derivatives of rhodanine-3-carboxyalkyl acidsDisruption of Myc-Max heterodimerization with improved cell-penetrating analogs of the small molecule 10074-G5.Development of Predictive QSAR Models of 4-Thiazolidinones Antitrypanosomal Activity using Modern Machine Learning Algorithms.Atropisomerism in 3-arylthiazolidine-2-thiones. A combined dynamic NMR and dynamic HPLC study.Recent developments with rhodanine as a scaffold for drug discovery.A green, multicomponent, regio- and stereo-selective 1,3-dipolar cycloaddition of azides and azomethine ylides generated in situ with bifunctional dipolarophiles using PEG-400.Synthesis of functionalized 5-substituted thiazolidine-2-thiones via adscititious xanthate-promoted radical cyclization of allyl(alkyl/aryl)dithiocarbamates.Structure activity relationship studies on rhodanines and derived enethiol inhibitors of metallo-β-lactamases.Synthesis, α-glucosidase inhibition and molecular docking studies of novel thiazolidine-2,4-dione or rhodanine derivativesChemical Instability and Promiscuity of Arylmethylidenepyrazolinone-Based MDMX Inhibitors
P2860
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P2860
Rhodanine as a scaffold in drug discovery: a critical review of its biological activities and mechanisms of target modulation.
description
2012 nî lūn-bûn
@nan
2012 թուականի Մայիսին հրատարակուած գիտական յօդուած
@hyw
2012 թվականի մայիսին հրատարակված գիտական հոդված
@hy
2012年の論文
@ja
2012年論文
@yue
2012年論文
@zh-hant
2012年論文
@zh-hk
2012年論文
@zh-mo
2012年論文
@zh-tw
2012年论文
@wuu
name
Rhodanine as a scaffold in dru ...... chanisms of target modulation.
@ast
Rhodanine as a scaffold in dru ...... chanisms of target modulation.
@en
Rhodanine as a scaffold in dru ...... chanisms of target modulation.
@nl
type
label
Rhodanine as a scaffold in dru ...... chanisms of target modulation.
@ast
Rhodanine as a scaffold in dru ...... chanisms of target modulation.
@en
Rhodanine as a scaffold in dru ...... chanisms of target modulation.
@nl
prefLabel
Rhodanine as a scaffold in dru ...... chanisms of target modulation.
@ast
Rhodanine as a scaffold in dru ...... chanisms of target modulation.
@en
Rhodanine as a scaffold in dru ...... chanisms of target modulation.
@nl
P2860
P1476
Rhodanine as a scaffold in dru ...... echanisms of target modulation
@en
P2093
Lucija Peterlin Mašič
Tihomir Tomašić
P2860
P304
P356
10.1517/17460441.2012.688743
P407
P577
2012-05-19T00:00:00Z