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Methods to Increase the Metabolic Stability of (18)F-RadiotracersBoronic Acid for the Traceless Delivery of Proteins into CellsCovalent Modifiers: A Chemical Perspective on the Reactivity of α,β-Unsaturated Carbonyls with Thiols via Hetero-Michael Addition ReactionsGypsogenin derivatives: an unexpected class of inhibitors of cholinesterases.Probing the carboxyester side chain in controlled deactivation (-)-δ(8)-tetrahydrocannabinols.Using click chemistry toward novel 1,2,3-triazole-linked dopamine D3 receptor ligands.A Resveratrol Analogue Promotes ERKMAPK-Dependent Stat3 Serine and Tyrosine Phosphorylation Alterations and Antitumor Effects In Vitro against Human Tumor Cells.Isolation and characterization of arylacetamide deacetylase in cynomolgus macaques.Mammalian alpha beta hydrolase domain (ABHD) proteins: Lipid metabolizing enzymes at the interface of cell signaling and energy metabolism.Monoclonal antibodies to human butyrylcholinesterase reactive with butyrylcholinesterase in animal plasma.Smart Mesoporous Nanomaterials for Antitumor Therapy.Nature as a source of metabolites with cholinesterase-inhibitory activity: an approach to Alzheimer's disease treatment.Phage therapy: eco-physiological pharmacology.Non-neuronal cholinergic system in airways and lung cancer susceptibility.Glycoengineering of Esterase Activity through Metabolic Flux-Based Modulation of Sialic Acid.Arylacetamide Deacetylase is Responsible for Activation of Prasugrel in Human and Dog.Enhancement of Curcumin Bioavailability Via the Prodrug Approach: Challenges and Prospects.Hexahydroquinolines are antimalarial candidates with potent blood-stage and transmission-blocking activity.Effect of Rifampin on the Disposition of Brivaracetam in Human Subjects: Further Insights into Brivaracetam Hydrolysis.Esterase phenotyping in human liver in vitro: specificity of carboxylesterase inhibitors.Absorption and cleavage of enalapril, a carboxyl ester prodrug, in the rat intestine: in vitro, in situ intestinal perfusion and portal vein cannulation models.New chemiluminescent substrates of paraoxonase 1 with improved specificity: synthesis and properties.Novel C-Ring-Hydroxy-Substituted Controlled Deactivation Cannabinergic Analogues.Human carboxylesterase 2: Studies on the role of glycosylation for enzymatic activity.Covalent inhibition of recombinant human carboxylesterase 1 and 2 and monoacylglycerol lipase by the carbamates JZL184 and URB597Use of 3-[(18)F]fluoropropanesulfonyl chloride as a prosthetic agent for the radiolabelling of amines: Investigation of precursor molecules, labelling conditions and enzymatic stability of the corresponding sulfonamidesDevelopment of a Novel Formulation That Improves Preclinical Bioavailability of Tenofovir Disoproxil Fumarate.Identification and Characterization of CINPA1 Metabolites Facilitates Structure-Activity Studies of the Constitutive Androstane Receptor.GRASr2 evaluation of aliphatic acyclic and alicyclic terpenoid tertiary alcohols and structurally related substances used as flavoring ingredients.Arylacetamide Deacetylase Is Involved in Vicagrel Bioactivation in Humans.Increased Biosynthetic Gene Dosage in a Genome-Reduced Defensive Bacterial Symbiont.Identification and optimization of soluble epoxide hydrolase inhibitors with dual potency towards fatty acid amide hydrolase.Metabolite profiling of carbamazepine and ibuprofen in Solea senegalensis bile using high-resolution mass spectrometry.Novel Genetic Variants in Carboxylesterase 1 Predict Severe Early-Onset Capecitabine-Related Toxicity.Metabolic Hydrolysis of Aromatic Amides in Selected Rat, Minipig, and Human In Vitro Systems.AADAC deacetylates PHENSynthetic cannabimimetic agents metabolized by carboxylesterases.Predominant contributions of carboxylesterase 1 and 2 in hydrolysis of anordrin in humans.A Novel Amino Lipid Series for mRNA Delivery: Improved Endosomal Escape and Sustained Pharmacology and Safety in Non-human Primates.Metabolism elucidation of BJ-B11 (a heat shock protein 90 inhibitor) by human liver microsomes: identification of main contributing enzymes.
P2860
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P2860
description
2012 nî lūn-bûn
@nan
2012 թուականի Յուլիսին հրատարակուած գիտական յօդուած
@hyw
2012 թվականի հուլիսին հրատարակված գիտական հոդված
@hy
2012年の論文
@ja
2012年論文
@yue
2012年論文
@zh-hant
2012年論文
@zh-hk
2012年論文
@zh-mo
2012年論文
@zh-tw
2012年论文
@wuu
name
The emerging role of human esterases.
@ast
The emerging role of human esterases.
@en
The emerging role of human esterases.
@nl
type
label
The emerging role of human esterases.
@ast
The emerging role of human esterases.
@en
The emerging role of human esterases.
@nl
prefLabel
The emerging role of human esterases.
@ast
The emerging role of human esterases.
@en
The emerging role of human esterases.
@nl
P1476
The emerging role of human esterases.
@en
P2093
Tatsuki Fukami
Tsuyoshi Yokoi
P304
P356
10.2133/DMPK.DMPK-12-RV-042
P577
2012-07-17T00:00:00Z