Covalent inhibition of recombinant human carboxylesterase 1 and 2 and monoacylglycerol lipase by the carbamates JZL184 and URB597
about
Metabolically Labile Fumarate Esters Impart Kinetic Selectivity to Irreversible InhibitorsIdentification of palmitoyl protein thioesterase 1 in human THP1 monocytes and macrophages and characterization of unique biochemical activities for this enzymeAcetylcholinesterase inhibitors: pharmacology and toxicology.Blocking of fatty acid amide hydrolase activity with PF-04457845 in human brain: a positron emission tomography study with the novel radioligand [(11)C]CURB.Effects of toxicologically relevant xenobiotics and the lipid-derived electrophile 4-hydroxynonenal on macrophage cholesterol efflux: silencing carboxylesterase 1 has paradoxical effects on cholesterol uptake and efflux.Interaction of the serine hydrolase KIAA1363 with organophosphorus agents: Evaluation of potency and kinetics.Simplified assays of lipolysis enzymes for drug discovery and specificity assessment of known inhibitors.Endocannabinoid hydrolases in avian HD11 macrophages identified by chemoproteomics: inactivation by small-molecule inhibitors and pathogen-induced downregulation of their activity.Identification and optimization of soluble epoxide hydrolase inhibitors with dual potency towards fatty acid amide hydrolase.Design and Potency of Dual Soluble Epoxide Hydrolase/Fatty Acid Amide Hydrolase Inhibitors
P2860
Q28817980-755E4E95-FBBA-4F7E-A6FE-1A6C741E6ECCQ33917127-3C74D44C-6D79-427A-82DE-CE6534510A28Q34381860-A0C1731B-A3B4-40B7-9EBC-B0636619A299Q36254356-83EB8A34-734A-4012-B667-8C148C030D93Q38953786-5C58DE8A-22A2-41FA-8C91-8E01538F6F5EQ41815378-2698243D-DD26-4780-AB76-AD09D4B7713BQ41906728-EEA3A9EE-DD49-4B52-8B78-7C1FCB9B6408Q47339481-8D50A639-97C0-4A9D-9A00-769ED402D02BQ47714123-E5AEE385-810A-4295-9DB0-A8FD30966D46Q58580945-14874605-87FF-426A-B61C-E742E26B8771
P2860
Covalent inhibition of recombinant human carboxylesterase 1 and 2 and monoacylglycerol lipase by the carbamates JZL184 and URB597
description
2012 nî lūn-bûn
@nan
2012年の論文
@ja
2012年論文
@yue
2012年論文
@zh-hant
2012年論文
@zh-hk
2012年論文
@zh-mo
2012年論文
@zh-tw
2012年论文
@wuu
2012年论文
@zh
2012年论文
@zh-cn
name
Covalent inhibition of recombi ...... e carbamates JZL184 and URB597
@en
type
label
Covalent inhibition of recombi ...... e carbamates JZL184 and URB597
@en
prefLabel
Covalent inhibition of recombi ...... e carbamates JZL184 and URB597
@en
P2093
P2860
P1476
Covalent inhibition of recombi ...... e carbamates JZL184 and URB597
@en
P2093
Abdolsamad Borazjani
J Allen Crow
Matthew K Ross
Victoria Bittles
P2860
P304
P356
10.1016/J.BCP.2012.08.017
P407
P577
2012-08-27T00:00:00Z