Structure-activity relationships in human Toll-like receptor 8-active 2,3-diamino-furo[2,3-c]pyridines.
about
Structure-Based Design of Novel Human Toll-like Receptor 8 AgonistsMulti-substituted 8-aminoimidazo[1,2-a]pyrazines by Groebke-Blackburn-Bienaymé reaction and their Hsp90 inhibitory activityVirtual Screening Approaches towards the Discovery of Toll-Like Receptor ModulatorsIdentification of Adjuvantic Activity of Amphotericin B in a Novel, Multiplexed, Poly-TLR/NLR High-Throughput Screen.Enrichment assessment of multiple virtual screening strategies for Toll-like receptor 8 agonists based on a maximal unbiased benchmarking data set.Human Toll-like receptor 8-selective agonistic activities in 1-alkyl-1H-benzimidazol-2-aminesDeterminants of activity at human Toll-like receptors 7 and 8: quantitative structure-activity relationship (QSAR) of diverse heterocyclic scaffolds.Structure-Based Design of Human TLR8-Specific Agonists with Augmented Potency and Adjuvanticity.Recent advances in development of imidazo[1,2-a]pyrazines: synthesis, reactivity and their biological applications.Groebke-Blackburn-Bienaymé multicomponent reaction: emerging chemistry for drug discovery.Exquisite selectivity for human toll-like receptor 8 in substituted furo[2,3-c]quinolines.Copper catalyzed synthesis of fused benzimidazolopyrazine derivatives via tandem benzimidazole formation/annulation of δ-alkynyl aldehyde.Small-molecule inhibition of TLR8 through stabilization of its resting state.Study on the agonists for the human Toll-like receptor-8 by molecular modeling.Syntheses of Human TLR8-Specific Small-Molecule Agonists.
P2860
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P2860
Structure-activity relationships in human Toll-like receptor 8-active 2,3-diamino-furo[2,3-c]pyridines.
description
2012 nî lūn-bûn
@nan
2012 թուականի Սեպտեմբերին հրատարակուած գիտական յօդուած
@hyw
2012 թվականի սեպտեմբերին հրատարակված գիտական հոդված
@hy
2012年の論文
@ja
2012年論文
@yue
2012年論文
@zh-hant
2012年論文
@zh-hk
2012年論文
@zh-mo
2012年論文
@zh-tw
2012年论文
@wuu
name
Structure-activity relationshi ...... -diamino-furo[2,3-c]pyridines.
@ast
Structure-activity relationshi ...... -diamino-furo[2,3-c]pyridines.
@en
Structure-activity relationshi ...... -diamino-furo[2,3-c]pyridines.
@nl
type
label
Structure-activity relationshi ...... -diamino-furo[2,3-c]pyridines.
@ast
Structure-activity relationshi ...... -diamino-furo[2,3-c]pyridines.
@en
Structure-activity relationshi ...... -diamino-furo[2,3-c]pyridines.
@nl
prefLabel
Structure-activity relationshi ...... -diamino-furo[2,3-c]pyridines.
@ast
Structure-activity relationshi ...... -diamino-furo[2,3-c]pyridines.
@en
Structure-activity relationshi ...... -diamino-furo[2,3-c]pyridines.
@nl
P2093
P2860
P356
P1476
Structure-activity relationshi ...... 3-diamino-furo[2,3-c]pyridines
@en
P2093
Katelyn J Serafin
Nikunj M Shukla
Rajalakshmi Balakrishna
Subbalakshmi S Malladi
Sunil A David
Victor W Day
P2860
P304
P356
10.1021/JM301066H
P407
P577
2012-09-07T00:00:00Z