Synthesis, biological activity, and crystal structure of potent nonnucleoside inhibitors of HIV-1 reverse transcriptase that retain activity against mutant forms of the enzyme.

Synthesis, biological activity, and crystal structure of potent nonnucleoside inhibitors of HIV-1 reverse transcriptase that retain activity against mutant forms of the enzyme.

Item
http://www.wikidata.org/entity/Q34674575
Fragment-based screening by X-ray crystallography, MS and isothermal titration calorimetry to identify PNMT (phenylethanolamine N-methyltransferase) inhibitorsIdentification of a 3-aminoimidazo[1,2-a]pyridine inhibitor of HIV-1 reverse transcriptase.SJP-L-5, a novel small-molecule compound, inhibits HIV-1 infection by blocking viral DNA nuclear entry.Human immunodeficiency virus reverse transcriptase: 25 years of research, drug discovery, and promise.2-(4-Meth-oxy-phen-yl)-1-phenyl-1H-benzimidazoleCombined Pd/C and Montmorillonite Catalysis for One-Pot Synthesis of Benzimidazoles.Comprehensive Review in Current Developments of Benzimidazole-Based Medicinal Chemistry.Novel fluorine-containing DAPY derivatives as potent HIV-1 NNRTIs: a patent evaluation of WO2014072419.Efficient aerobic oxidative synthesis of 2-substituted benzoxazoles, benzothiazoles, and benzimidazoles catalyzed by 4-methoxy-TEMPO.One-pot strategy of copper-catalyzed synthesis of 1,2-disubstituted benzimidazoles.Novel Mcl-1/Bcl-2 dual inhibitors created by the structure-based hybridization of drug-divided building blocks and a fragment deconstructed from a known two-face BH3 mimetic.From TIBO to Rilpivirine: The Chronicle of the Discovery of the Ideal Nonnucleoside Reverse Transcriptase Inhibitor
P2860

Synthesis, biological activity, and crystal structure of potent nonnucleoside inhibitors of HIV-1 reverse transcriptase that retain activity against mutant forms of the enzyme.

Item
http://www.wikidata.org/entity/Q34674575
description
2007 nî lūn-bûn
@nan
2007 թուականի Յուլիսին հրատարակուած գիտական յօդուած
@hyw
2007 թվականի հուլիսին հրատարակված գիտական հոդված
@hy
2007年の論文
@ja
2007年論文
@yue
2007年論文
@zh-hant
2007年論文
@zh-hk
2007年論文
@zh-mo
2007年論文
@zh-tw
2007年论文
@wuu
name
Synthesis, biological activity ...... st mutant forms of the enzyme.
@ast
Synthesis, biological activity ...... st mutant forms of the enzyme.
@en
Synthesis, biological activity ...... st mutant forms of the enzyme.
@nl
type
label
Synthesis, biological activity ...... st mutant forms of the enzyme.
@ast
Synthesis, biological activity ...... st mutant forms of the enzyme.
@en
Synthesis, biological activity ...... st mutant forms of the enzyme.
@nl
prefLabel
Synthesis, biological activity ...... st mutant forms of the enzyme.
@ast
Synthesis, biological activity ...... st mutant forms of the enzyme.
@en
Synthesis, biological activity ...... st mutant forms of the enzyme.
@nl
P1433
P1476
P2093
P2860
P304
P31
P356
P407
P433
P478
P50
P577
P5875
P698
P921
P932
P356
P1433
P1476
Synthesis, biological activity ...... st mutant forms of the enzyme.
@en
P2093
P2860
P304
P31
P356
P407
P433
P478
P50
P577
P5875
P698
P921
P932