Screen of pseudopeptidic inhibitors of human sirtuins 1-3: two lead compounds with antiproliferative effects in cancer cells.
about
Sirtuin functions and modulation: from chemistry to the clinicDevelopment and characterization of 3-(benzylsulfonamido)benzamides as potent and selective SIRT2 inhibitorsDual Genetic Encoding of Acetyl-lysine and Non-deacetylatable Thioacetyl-lysine Mediated by Flexizyme[Dual genetic encoding of acetyl-lysine and non-deacetylatablethioacetyl-lysine mediated by flexizyme].The sirtuin class of histone deacetylases: regulation and roles in lipid metabolism.Sirtuin inhibitors as anticancer agents.BET Inhibition Upregulates SIRT1 and Alleviates Inflammatory Responses.Endothioxopeptides: A conformational overview.The discovery of a highly selective 5,6,7,8-tetrahydrobenzo[4,5]thieno[2,3-d]pyrimidin-4(3H)-one SIRT2 inhibitor that is neuroprotective in an in vitro Parkinson's disease model.The Current State of NAD(+) -Dependent Histone Deacetylases (Sirtuins) as Novel Therapeutic Targets.Potent mechanism-based sirtuin-2-selective inhibition by an in situ-generated occupant of the substrate-binding site, "selectivity pocket" and NAD+-binding site.Thienopyrimidinone Based Sirtuin-2 (SIRT2)-Selective Inhibitors Bind in the Ligand Induced Selectivity Pocket.
P2860
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P2860
Screen of pseudopeptidic inhibitors of human sirtuins 1-3: two lead compounds with antiproliferative effects in cancer cells.
description
2013 nî lūn-bûn
@nan
2013 թուականի Օգոստոսին հրատարակուած գիտական յօդուած
@hyw
2013 թվականի օգոստոսին հրատարակված գիտական հոդված
@hy
2013年の論文
@ja
2013年論文
@yue
2013年論文
@zh-hant
2013年論文
@zh-hk
2013年論文
@zh-mo
2013年論文
@zh-tw
2013年论文
@wuu
name
Screen of pseudopeptidic inhib ...... ative effects in cancer cells.
@ast
Screen of pseudopeptidic inhib ...... ative effects in cancer cells.
@en
Screen of pseudopeptidic inhib ...... ative effects in cancer cells.
@nl
type
label
Screen of pseudopeptidic inhib ...... ative effects in cancer cells.
@ast
Screen of pseudopeptidic inhib ...... ative effects in cancer cells.
@en
Screen of pseudopeptidic inhib ...... ative effects in cancer cells.
@nl
prefLabel
Screen of pseudopeptidic inhib ...... ative effects in cancer cells.
@ast
Screen of pseudopeptidic inhib ...... ative effects in cancer cells.
@en
Screen of pseudopeptidic inhib ...... ative effects in cancer cells.
@nl
P2093
P50
P356
P1476
Screen of pseudopeptidic inhib ...... ative effects in cancer cells.
@en
P2093
Elina M Jarho
Heikki S Salo
Laura Tolvanen
Tiina Suuronen
P304
P356
10.1021/JM400438K
P407
P577
2013-08-22T00:00:00Z