Binding sites for bilobalide, diltiazem, ginkgolide, and picrotoxinin at the 5-HT3 receptor.
about
Applying linear and non-linear methods for parallel prediction of volume of distribution and fraction of unbound drugThe Concise Guide to PHARMACOLOGY 2013/14: ligand-gated ion channels.Azemiopsin from Azemiops feae viper venom, a novel polypeptide ligand of nicotinic acetylcholine receptor.Neuroprotective effects of bilobalide on cerebral ischemia and reperfusion injury are associated with inhibition of pro-inflammatory mediator production and down-regulation of JNK1/2 and p38 MAPK activation.Phenylalanine in the pore of the Erwinia ligand-gated ion channel modulates picrotoxinin potency but not receptor functionA single amino acid determines the toxicity of Ginkgo biloba extracts.VUF10166, a novel compound with differing activities at 5-HT₃A and 5-HT₃AB receptors.The pharmacological profile of ELIC, a prokaryotic GABA-gated receptorMixed antagonistic effects of the ginkgolides at recombinant human ρ1 GABAC receptorsA single channel mutation alters agonist efficacy at 5-HT3A and 5-HT3AB receptors.Noncompetitive Inhibition of 5-HT3 Receptors by Citral, Linalool, and Eucalyptol Revealed by Nonlinear Mixed-Effects Modeling.Discriminating between 5-HT₃A and 5-HT₃AB receptorsCysteine modification reveals which subunits form the ligand binding site in human heteromeric 5-HT3AB receptors.Cys-loop receptor channel blockers also block GLIC.Structure-activity relationships of quinoxaline-based 5-HT3A and 5-HT3AB receptor-selective ligands.5-HT3 Receptor Brain-Type B-Subunits are Differentially Expressed in Heterologous Systems.Probing residues in the pore-forming (M2) domain of the Cys-loop receptor homologue GLIC reveals some unusual features.Identification of Glycyrrhiza as the rikkunshito constituent with the highest antagonistic potential on heterologously expressed 5-HT3A receptors due to the action of flavonoids.A golden approach to ion channel inhibitionAn atypical residue in the pore of Varroa destructor GABA-activated RDL receptors affects picrotoxin block and thymol modulationThe L-type voltage-gated calcium channel CaV1.2 mediates fear extinction and modulates synaptic tone in the lateral amygdala.Subunit-dependent inhibition and potentiation of 5-HT3 receptor by the anticancer drug, topotecan.
P2860
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P2860
Binding sites for bilobalide, diltiazem, ginkgolide, and picrotoxinin at the 5-HT3 receptor.
description
2011 nî lūn-bûn
@nan
2011 թուականի Ապրիլին հրատարակուած գիտական յօդուած
@hyw
2011 թվականի ապրիլին հրատարակված գիտական հոդված
@hy
2011年の論文
@ja
2011年論文
@yue
2011年論文
@zh-hant
2011年論文
@zh-hk
2011年論文
@zh-mo
2011年論文
@zh-tw
2011年论文
@wuu
name
Binding sites for bilobalide, ...... toxinin at the 5-HT3 receptor.
@ast
Binding sites for bilobalide, ...... toxinin at the 5-HT3 receptor.
@en
type
label
Binding sites for bilobalide, ...... toxinin at the 5-HT3 receptor.
@ast
Binding sites for bilobalide, ...... toxinin at the 5-HT3 receptor.
@en
prefLabel
Binding sites for bilobalide, ...... toxinin at the 5-HT3 receptor.
@ast
Binding sites for bilobalide, ...... toxinin at the 5-HT3 receptor.
@en
P2093
P2860
P356
P1476
Binding sites for bilobalide, ...... toxinin at the 5-HT3 receptor.
@en
P2093
A J Thompson
S C R Lummis
P2860
P304
P356
10.1124/MOL.111.071415
P577
2011-04-19T00:00:00Z