Functional reconstitution of Haemonchus contortus acetylcholine receptors in Xenopus oocytes provides mechanistic insights into levamisole resistance.
about
The genome and transcriptome of Haemonchus contortus, a key model parasite for drug and vaccine discoveryIs anthelmintic resistance a concern for the control of human soil-transmitted helminths?Principles of agonist recognition in Cys-loop receptorsFunctional Characterization of a Novel Class of Morantel-Sensitive Acetylcholine Receptors in NematodesRecent Duplication and Functional Divergence in Parasitic Nematode Levamisole-Sensitive Acetylcholine ReceptorsExpression of nicotinic acetylcholine receptor subunits from parasitic nematodes in Caenorhabditis elegans.Genomic introgression mapping of field-derived multiple-anthelmintic resistance in Teladorsagia circumcinctaPositive modulation of a Cys-loop acetylcholine receptor by an auxiliary transmembrane subunit.Xenopus laevis RIC-3 enhances the functional expression of the C. elegans homomeric nicotinic receptor, ACR-16, in Xenopus oocytes.The Conqueror Worm: recent advances with cholinergic anthelmintics and techniques excite research for better therapeutic drugs.Recent advances in candidate-gene and whole-genome approaches to the discovery of anthelmintic resistance markers and the description of drug/receptor interactions.Computational cloning of drug target genes of a parasitic nematode, Oesophagostomum dentatum.Tribendimidine: mode of action and nAChR subtype selectivity in Ascaris and OesophagostomumHeterologous Expression in Remodeled C. elegans: A Platform for Monoaminergic Agonist Identification and Anthelmintic Screening.Expression of five acetylcholine receptor subunit genes in Brugia malayi adult wormsSelective effect of the anthelmintic bephenium on Haemonchus contortus levamisole-sensitive acetylcholine receptors.Levamisole receptors: a second awakening.The Ascaris suum nicotinic receptor, ACR-16, as a drug target: Four novel negative allosteric modulators from virtual screening.Whole-cell patch-clamp recording of nicotinic acetylcholine receptors in adult Brugia malayi muscle.Pharmacological profile of Ascaris suum ACR-16, a new homomeric nicotinic acetylcholine receptor widely distributed in Ascaris tissuesAcetylcholine receptor subunit and P-glycoprotein transcription patterns in levamisole-susceptible and -resistant Haemonchus contortus.Parasite neuropeptide biology: Seeding rational drug target selection?P-glycoproteins and other multidrug resistance transporters in the pharmacology of anthelmintics: Prospects for reversing transport-dependent anthelmintic resistance.Ion channels and receptor as targets for the control of parasitic nematodes.Investigation of acetylcholine receptor diversity in a nematode parasite leads to characterization of tribendimidine- and derquantel-sensitive nAChRs.Impacts of chronic low-level nicotine exposure on Caenorhabditis elegans reproduction: identification of novel gene targets.Transcriptomic evaluation of the nicotinic acetylcholine receptor pathway in levamisole-resistant and -sensitive Oesophagostomum dentatum.The evolution of pentameric ligand-gated ion-channels and the changing family of anthelmintic drug targets.Acetylcholinesterase and Nicotinic Acetylcholine Receptors in Schistosomes and Other Parasitic Helminths.Drug-efflux and target-site gene expression patterns in Haemonchus contortus larvae able to survive increasing concentrations of levamisole in vitroMonepantel is a non-competitive antagonist of nicotinic acetylcholine receptors from Ascaris suum and Oesophagostomum dentatum.Deciphering the molecular determinants of cholinergic anthelmintic sensitivity in nematodes: When novel functional validation approaches highlight major differences between the model Caenorhabditis elegans and parasitic species.
P2860
Q21183984-341EBB73-C091-45C0-9DB3-1205950413DBQ26991607-A1B58958-1739-4819-82DD-FCF0199B0672Q28239408-2B50A9F4-1DE2-42DF-9155-66AE4623975BQ28551220-A4B1E92A-7B0C-40BA-BF5B-2D2D9ADC2E75Q28552649-E4077878-63DC-495D-858D-6B079B08E6ADQ30702478-D22A65C5-D05A-444D-BAC7-BA5EEE3CC620Q33897920-9DBFC5D8-65FC-46D3-9AB3-F9BB8454A136Q34295982-11F1D303-6E9F-4BEA-A954-75B651E00924Q34299221-6303326A-BB7C-4594-8781-5CD2D75B9491Q34587731-A2F9331A-6991-46A9-924A-4DBD13666551Q34705912-8E695F20-2BD8-4AD1-9999-33E8FE923CDFQ34774856-CF72DF35-EC21-4F0E-BCEF-E8727069066FQ35101636-91F50D53-4717-47D7-8974-9ECED73633ADQ35557727-B4649BD3-B17D-4EB8-A420-03B2B4E8E59CQ35864932-43AFEFED-E1D0-458E-AB18-B5CA90031D9DQ35995069-09B15B6C-6321-46E9-8BFD-381602EB22EAQ36044037-99F5327A-53A8-455C-8202-257C351F9C2CQ36724064-6C4AEDE8-F189-4223-A60F-178172EEA087Q37097877-05DDB733-83DE-4820-ADA9-46DC88E058E7Q37123991-7B63B2DE-FF94-4585-8046-17F431FB0FFEQ37390593-B89CE8A2-A8EC-42D3-8A12-F889123B694AQ37390597-41D78A82-6A70-418D-8D58-86CA477FA9A5Q37390601-2C867BD1-8A81-42B2-B724-EB9F63B52A17Q37501925-F28AF3C0-0C68-4DDC-B73F-09BFE071F5ABQ37533979-8C79F684-B140-4769-84AF-3C5699805CEAQ37603263-9C99B149-AAFB-451D-AF5D-C69B67FAD4AFQ37712241-D4624C2C-772E-429A-B42D-65EB65951412Q38263700-695CC201-8FBE-4EF8-A2D2-AD83B51C9B38Q40046503-04001193-504C-4E52-8928-324E0B6699E2Q41986089-6DEFCCAE-9946-400B-8CC0-996803FBDA22Q48502792-382BE745-8AC8-4130-A4AD-73248AB190D9Q54998446-FCDDC6B1-5850-468E-885A-A4BB51F595C5
P2860
Functional reconstitution of Haemonchus contortus acetylcholine receptors in Xenopus oocytes provides mechanistic insights into levamisole resistance.
description
2011 nî lūn-bûn
@nan
2011年の論文
@ja
2011年論文
@yue
2011年論文
@zh-hant
2011年論文
@zh-hk
2011年論文
@zh-mo
2011年論文
@zh-tw
2011年论文
@wuu
2011年论文
@zh
2011年论文
@zh-cn
name
Functional reconstitution of H ...... ts into levamisole resistance.
@ast
Functional reconstitution of H ...... ts into levamisole resistance.
@en
type
label
Functional reconstitution of H ...... ts into levamisole resistance.
@ast
Functional reconstitution of H ...... ts into levamisole resistance.
@en
prefLabel
Functional reconstitution of H ...... ts into levamisole resistance.
@ast
Functional reconstitution of H ...... ts into levamisole resistance.
@en
P2093
P2860
P50
P1476
Functional reconstitution of H ...... hts into levamisole resistance
@en
P2093
P2860
P304
P356
10.1111/J.1476-5381.2011.01420.X
P407
P577
2011-11-01T00:00:00Z